Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
JPNUKJAOPRHHRY 8.9 Ki 5
XRIVGYHVHPSIIW 8.9 Ki 5
UBFYWPOOPLWTOY 8.9 Ki 2
CKEZLGKKMUHEMS 8.8 IC50 2
FAEVMLINNNVLLK 8.8 Ki 5
IJGXBJUJDSODSN 8.8 Ki 4
WPYTXBRSQCLTAR 8.8 IC50 2
ZAGVNQCMOLWFKV 8.8 Ki 5
PYSCVJMLJRHJGJ 8.8 Ki 2
UBFPRQOOAXMTBD 8.8 IC50 6
LPKHNHHBGJUJHL 8.8 Ki 2
NGYNSMZIHJNHSS 8.8 Ki 2
AQYPBNGIIYVIBQ 8.8 Ki 5
ILLGYRJAYAAAEW 8.8 Ki 3
JASZEBXICKBENQ 8.8 Ki 4
YJYPZLAZNIGNRP 8.8 Ki 3
CRCWSASAEVRBQR 8.8 Ki 2
XVOITFWFESABRI 8.8 Ki 4
ODQRKAFUQFOHEX 8.7 Ki 4
CLRANNZHQRADST 8.7 IC50 2
GKNSLBAHDKWDHQ 8.7 Ki 5
HCZNYXWSHKDVMC 8.7 Ki 2
ILEWLUJOKLLBMF 8.7 Ki 7
JBOVXXZNZSULJJ 8.7 IC50 2
JHFTWXCZLKAESI 8.7 Ki 2
NGGVRPGLGXDGKP 8.7 Ki 7
OVRHNZFXULSZGO 8.7 Ki 2
PSHDKMKDEJGTHJ 8.7 Ki 5
WLPPBIMGKKVATA 8.7 IC50 2
PWXQAVZNBKKQOF 8.7 Ki 7
UEQZFAGVRGWPDK 8.7 Ki 3
XKGJHXYHHLQEGC 8.7 Ki 5
XXKYVKOMLITFKH 8.7 Ki 2
YWDRNTZRCJXPPD 8.7 Ki 2
CSWXXYOKFXHTOD 8.7 IC50 2
VKUPFPYBQLXLIG 8.7 IC50 2
ACPHUHSYZGYUCK 8.6 Ki 5
YLCDIBDYBLQAJS 8.6 Ki 4
YLTFIHQASWBABS 8.6 Ki 2
MJRZXRNJFQLHHY 8.6 IC50 2
SIPSUTQRUBWRRD 8.6 IC50 2
SWPVFHZSTTYORI 8.6 IC50 5
BMELFMSHGRMUAH 8.6 Ki 2
CFWKQRTXGKVATK 8.6 Ki 2
XJHYAVIQMMKYJG 8.6 IC50 2
CHUVPNWRFUBJRL 8.6 Ki 5
DGINADWRRXVFLH 8.6 IC50 2
OIDZIVZCMGAXHN 8.6 Ki 2
FIZHAHHNRMPEKR 8.5 Ki 4
ISYFVYGWOGOQMZ 8.5 Ki 2
2D structure