Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
PDPSDBUFNKLMBE 9.2 IC50 2
DEXLAAAKAUMETM 9.2 Ki 5
OHTDTNHLFFCQRH 9.2 Ki 5
PMQMQOADOYNRNP 9.2 Ki 5
FRXNJQHCVWNOGI 9.2 IC50 2
GAGCCMIPRTXYNT 9.2 IC50 2
DNTSAGFCYYBUKZ 9.2 Ki 5
GTVWKLSULFFQST 9.2 Ki 7
YCKUJRLTYLJWTR 9.2 Ki 5
KFULFWHCQIMTLB 9.1 Ki 4
LPYOFVQCAYSFSJ 9.1 IC50 6
MUAAOAJMVIAASD 9.1 Ki 2
ZMRZCVHPEQNWCW 9.1 Ki 2
GEEFPQBPVBFCSD 9.1 Ki 2
ISACHQOCISQFPP 9.1 Ki 4
KEJDQVGYGBHLMC 9.1 Ki 4
RLPOPCNSEITQNR 9.1 Ki 4
CGMWYBOZPGNPIF 9.1 Ki 4
UGNNTIXQGYYUAP 9.1 IC50 2
WPVQUWLESAWSRM 9.1 IC50 2
APYCQWZCHZQKRW 9.1 IC50 2
DMDHFLXQSOBORU 9.1 Ki 5
GIUMMCXYLUQIND 9.1 Ki 5
LSPFRPGGOBZZFJ 9.0 Ki 2
BXQVWZDNOZKPLA 9.0 Ki 2
AQYPBNGIIYVIBQ 9.0 Ki 5
FAEVMLINNNVLLK 9.0 Ki 5
HFALPZZGNQXIMP 9.0 Ki 5
HFIMLFRJUJSWHZ 9.0 Ki 5
INYNWEUTASDACG 9.0 Ki 5
JRNYLCIPPWHNEJ 9.0 IC50 2
KPHRNXIFUJLFNL 9.0 Ki 5
SHALYUZFJLUFSL 9.0 IC50 2
SJGHGXWQPNNDCN 9.0 Ki 5
SKFPODQWUBSOEM 9.0 Ki 5
TWVKXXKMLUVNDJ 9.0 Ki 5
YMXSEXVSDUSENY 9.0 Ki 2
ACHWGHFEAPJMKT 9.0 Ki 5
AQYPBNGIIYVIBQ 9.0 Ki 5
CZZTUVCSFLVVCL 9.0 Ki 2
HXLVTGLHDULKSB 9.0 Ki 2
KUPJKPMGKUDEHS 9.0 Ki 2
SGNXVBOIDPPRJJ 9.0 Ki 2
UCMCIMRDJCGRNT 9.0 IC50 4
HCZDWLWWAVVIPY 8.9 Ki 2
ZTSSUVKQGBVRTE 8.9 Ki 2
PUMYSIXHQPYXGX 8.9 Ki 4
QBXBOZRRJVJSKZ 8.9 Ki 2
GQUWFILFBVDMRP 8.9 IC50 2
IZXOINQUSUGYPF 8.9 Ki 3
2D structure