Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
SLRAKVICRDZWAA 9.7 Ki 5
XBSNMYAFJJSQQL 9.7 Ki 2
ZLLCEWCZDFPICU 9.7 Ki 5
ZLLCEWCZDFPICU 9.7 Ki 5
ZNRNCCOAWBUSNP 9.7 Ki 4
GDSORCYTZJIZHU 9.7 Ki 4
OCEAINWYIRTVGD 9.6 Ki 5
VJEHPMOIYSUGSJ 9.6 Ki 2
AIARDFWQNXMLKK 9.6 Ki 2
LYGZRGMHPFAAMR 9.6 Ki 7
BACMDOCEIHERJI 9.6 Ki 3
CRXFCGUGNWJSEY 9.6 Ki 5
ANJTVLIZGCUXLD 9.6 Ki 9
KMIROODCYQMZLK 9.6 Ki 4
NNEPQECWOJJCPU 9.6 Ki 2
BEBIEORUESJWFE 9.5 Ki 5
DEXLAAAKAUMETM 9.5 Ki 5
DEXLAAAKAUMETM 9.5 Ki 5
KTCKWEYGXKJYMD 9.5 Ki 2
NHSPZGBYUPGTML 9.5 Ki 2
URCPIVZAKGXXGX 9.5 IC50 5
YSVOMDFBWJGXEL 9.5 Ki 5
ZLLCEWCZDFPICU 9.5 Ki 5
SOBKRFVVZYOGEO 9.5 Ki 2
RNOBTWYQAWEZHH 9.5 Ki 2
SGNXVBOIDPPRJJ 9.5 Ki 3
CRXFCGUGNWJSEY 9.5 Ki 5
BVMMXDPNJVFASA 9.4 Ki 2
LYMBELAAKZROPC 9.4 Ki 4
WBYFNWHZLPPQST 9.4 Ki 3
APBRBJOIYDBKFZ 9.4 Ki 2
BCTMPICFFTZGMY 9.4 IC50 2
RLSQXMJPNPUPPZ 9.4 Ki 2
BEXHXBAKDDOWBF 9.4 Ki 5
CRPBMTGSCRKOBR 9.4 Ki 5
GFPKENYJHPZLJI 9.4 Ki 2
IMWUFTIDVKJBTJ 9.4 Ki 5
PMMKTOLCURGBKI 9.4 Ki 4
PQBYYZBQJKBZMS 9.4 Ki 5
QCSSDCOJCQOKNU 9.4 Ki 5
HYDLTSOVXCUHPA 9.4 Ki 5
VKYSIJWKGXVHKX 9.4 Ki 2
RKHOYJFLFFRBNN 9.3 IC50 2
JKJZPYHBDCLWAB 9.3 Ki 2
LZJKYCFNHCYHCM 9.3 Ki 8
VHNSVCKCMBYGSB 9.3 Ki 5
WBRKKKJHXQZXEM 9.3 Ki 2
IMNMXRIDDYENFD 9.3 Ki 2
JGOKWXDQJRLPLM 9.3 Kd 2
GZAHUQFGFBFMCD 9.3 Ki 2
2D structure