Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
KKHBYNBHPMWTCF 6.2 Ki 3
RTEIKCPHPAQRML 6.2 Ki 2
UAVBXTCRHQYQIA 6.2 Ki 3
VWRPUTHGEXQRJZ 6.2 Ki 3
WXVSPYOOFCCEII 6.2 Ki 2
MLWYWGHZOHABMH 6.2 Ki 3
ZRCMYKLGYHVJGO 6.2 Ki 5
KJKJEMGOLPUHLS 6.2 IC50 2
ZYRONZISKSSHFA 6.2 IC50 2
MTCUAOILFDZKCO 6.2 Ki 4
QLOHOGRMRUDDPM 6.2 IC50 2
HMBUBSLJZZWVMM 6.2 Ki 2
VJEPFPRUUZASOL 6.2 Ki 5
OQFNODATXJBYQO 6.2 Ki 3
ALGQHHHCUISTSF 6.1 Ki 3
UFURGWJSEGJTTD 6.1 Ki 2
YWTYJOPNNQFBPC 6.1 Ki 2
QYIIVMFJYKZTIQ 6.1 Ki 4
TVQVEBXIMQEOQV 6.1 Ki 3
TZWVPYLQJDFQHL 6.1 Ki 5
XQZOCCXVRTXGTP 6.1 Ki 2
YRSRVRMUNDNIIH 6.1 Ki 3
FBFVECUFQXIPMF 6.1 Ki 3
JIGWWGDIEUWCOR 6.1 Ki 5
OIRQDWMLNIFQQH 6.1 Ki 3
UXFGZUGBPVWQSE 6.1 Ki 2
OHBUTCGNMVYVRF 6.1 IC50 2
UEHARNLMUOFGOF 6.1 IC50 3
XZMYNLLVUGBWFQ 6.1 Ki 2
NXYMRNPNBDPMMA 6.1 Ki 2
SLALSTOEQACNCW 6.1 Ki 3
SLDFYFBUCMPAFI 6.1 Ki 2
BLOYCIJJVGNWOB 6.0 Ki 2
CVJIJXSIQBMJHS 6.0 Ki 3
FZZUWACJRQRLAZ 6.0 Ki 3
IKXYPVOSZVQOPI 6.0 Ki 3
KFVYJNNGAANKPZ 6.0 Ki 3
RCCDDPHPJBBTOH 6.0 Ki 4
RPYCUDHNQUMCME 6.0 Ki 3
BNXKZZZGHZDNKA 6.0 Ki 2
FGUCOPALAZXICJ 6.0 Ki 2
JFJZZMVDLULRGK 6.0 Ki 3
GPCVUHGDQJVKPL 6.0 Ki 2
BQNSBENKJCLJGN 6.0 IC50 2
IBFLDAUDRHDONN 6.0 Ki 2
TTYPEICBBIVUBR 6.0 Ki 3
AJTVQZWUKUPHIP 6.0 IC50 3
DBHHVOXBHXZBFC 6.0 Ki 3
HSIBGVUMFOSJPD 6.0 IC50 6
ICKPJMDBIACNSE 6.0 Ki 3
2D structure