Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
BFWLEZJNBVFENH 6.7 Ki 2
DMBSWJMVDSGAIT 6.7 Ki 3
DTUYFIYHCUBCJI 6.7 IC50 3
FLASSHOGJKRSGA 6.7 Ki 2
FPPMNAOECAYTAK 6.7 Ki 2
HTBCXNBZJPZOBH 6.7 Ki 3
MQWQCNHPYKVXNY 6.7 Ki 2
UOODLUFDPIXJIH 6.7 Ki 2
ZKWHETNMJXBGTO 6.7 Ki 5
ZWCVNJVVVNDHTO 6.7 Ki 3
BADPXOSJBUEVTR 6.7 IC50 3
BADPXOSJBUEVTR 6.7 IC50 2
SOMFWHZONIFICL 6.7 Ki 2
ADPGBLDMLCUZBX 6.7 Ki 5
ZKWHETNMJXBGTO 6.7 Ki 3
ZVCAGLIRHWFFLH 6.7 Ki 2
MYGGRYSOINDCAP 6.6 Ki 3
MYGGRYSOINDCAP 6.6 Ki 5
QWFZPQDYBCZVNF 6.6 Ki 2
SKKUGGANPAFLLZ 6.6 IC50 2
UJPISKKZQVLXEM 6.6 Ki 3
CREADRXFMNTHBO 6.6 IC50 2
PZQYPZNWIIVXRR 6.6 Ki 2
KPURMDWMUNJNJZ 6.6 Ki 2
MTRLPURDJAKESO 6.6 IC50 2
ORNGHPVNFVLRNV 6.6 Ki 4
WITLOMKPGROHOE 6.6 Ki 4
WXTQMACZCSXJTB 6.6 Ki 4
CCEBJZRLEVFTNS 6.6 IC50 4
CEIOZCMVGWULLM 6.6 Ki 2
WGTASENVNYJZBK 6.6 Ki 7
CKRXLDDIUCBOSQ 6.6 Ki 2
QSGXLBLODQIGSD 6.6 Ki 2
BGFXQHQMJCEQEA 6.5 IC50 2
MZZNJWVIWBAYRS 6.5 IC50 2
IJYFQAUVWBRZIV 6.5 Ki 3
ZBIKLRAGWSOQHD 6.5 IC50 2
MGCYWLIOYRXTDE 6.5 IC50 4
MYRHBCKCPROFGA 6.5 IC50 2
BGQXOWCDCVCZJN 6.5 Ki 2
SZRDMKGSPWOQFL 6.5 Ki 2
DMDCNPUUEFFDRN 6.5 Ki 2
YVMHTPXPXBMVRH 6.5 Ki 2
GLDKDAVDPFANSF 6.5 Ki 3
HUGVWLBFJCKUSU 6.5 Ki 3
NIYRJBGYQWFLAO 6.5 Ki 2
PYSCVJMLJRHJGJ 6.5 Ki 4
VTNUIOCYBBUEHK 6.5 Ki 5
CWYMBKHGVCNXNE 6.5 Ki 2
RFLDYHWWEJNDMO 6.5 Ki 4
2D structure