Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
ADQYVAWNTXPENQ 7.0 IC50 3
DCWKRPJLVIHGCZ 7.0 IC50 2
HXWNIHVLKOKITO 7.0 Ki 2
NZGNBOYHACXVNU 7.0 Ki 3
HZQBHNQELXWIPY 7.0 Ki 2
ULUVSICUEWOINW 7.0 Ki 5
UAFJMITWUKBNEN 7.0 IC50 5
BWIJRTTXRLQRFV 7.0 Ki 2
CEVPPNAINXEGSH 7.0 IC50 2
CRHHYTWGPWXCHF 7.0 Ki 2
XMOYAAVIEIXMBH 7.0 Ki 2
WBAIXNUCEGCLDC 7.0 Ki 2
XLTANAWLDBYGFU 7.0 IC50 2
YSSBTWFASLVAGY 7.0 IC50 5
ZRQYLGIDTXZHEU 6.9 Ki 2
ATULJSMRIAVHMJ 6.9 IC50 2
BGRDESOBNOVWPL 6.9 Ki 5
GSPNWTCHDVQYCA 6.9 Ki 2
KHRMJWYROCGIKU 6.9 Ki 3
OHOAHMFSJUWQMW 6.9 Ki 2
CZYVZKBXPYWXIG 6.9 Ki 2
JFPXLNSBLNDHFH 6.9 IC50 4
PKIKIQOOXGRVIT 6.9 Ki 5
FRKHHIZFRUBRFE 6.9 Ki 2
CAYMRNQWSQYOLB 6.8 Ki 4
CAYMRNQWSQYOLB 6.8 Ki 2
OCKIPDMKGPYYJS 6.8 Ki 4
OFTPVHUJNOOXJO 6.8 Ki 3
WXTQMACZCSXJTB 6.8 Ki 4
XSJCLLVXAXKDRO 6.8 Ki 2
IOHRCEONZVRYRI 6.8 IC50 2
NQSGGIDOQYCFCP 6.8 Ki 5
XUZOLWBRVIFEEI 6.8 Ki 2
BZXBTMGFASFGQD 6.8 Ki 2
GFZPTQHNFIWYND 6.8 Ki 2
JWEOQIUDCVEFPL 6.8 Ki 2
MOCURCBRVYTAME 6.8 Ki 4
OXKRFEWMSWPKKV 6.8 Ki 3
AOOOIKZSTAKHBL 6.8 Ki 2
GOLBTOIFBMVFTQ 6.8 IC50 2
NRUGCGUIOWHUGI 6.8 IC50 2
SYCMNXTXRHUPAZ 6.8 IC50 2
STOHKMQGYFFHMS 6.8 Ki 2
IXIGRKFDMBWCOA 6.8 Ki 3
CHQFGLQUINKUJZ 6.7 IC50 2
OVRZSDRDBJDKBF 6.7 IC50 2
ZBCPFWOYXGGVNU 6.7 Ki 2
FDNXWEUROWLDDO 6.7 Ki 2
GHJPZQCAVQYABA 6.7 IC50 2
VBUZMQUXIQZALI 6.7 IC50 2
2D structure