Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
FQIJPHXWIONJLF 7.3 IC50 2
LFBLWBXTTPQJNY 7.3 Ki 2
PKQIBCQLDRUHEO 7.3 IC50 2
RPYWXZCFYPVCNQ 7.3 Ki 3
VQUBBGRWUMHAJX 7.3 IC50 2
HSPGCGUPFQHASA 7.3 Ki 2
SCQZDZCGZMOONT 7.3 Ki 2
XEOOLDLJXYEALJ 7.3 Ki 3
ZAVZYZZLAYQHQP 7.3 Ki 2
DYJPSVCASDBOSA 7.2 Ki 4
VMEDIUSDIYRUSA 7.2 IC50 10
DFVICVZMQQSUPU 7.2 Ki 2
JFWOCEJLRQNSEH 7.2 IC50 3
PPNVCWLCUGAHAI 7.2 IC50 2
TVQVEBXIMQEOQV 7.2 IC50 4
VIWKHXNVEIOPSC 7.2 IC50 10
AMOKJMKEFDPTPN 7.2 IC50 7
FLOMZNVQFVMELR 7.2 Ki 2
QVUMHMHDZSGOQN 7.2 Ki 2
RJANNBFEAICXLW 7.2 IC50 2
CSSMYCLAVGYSEW 7.2 Ki 2
KIUXROKMRBBOBZ 7.2 Ki 2
DYUZUWODHHENIO 7.2 Ki 2
UDGISDAHRCDXMV 7.2 IC50 6
CZWUYUYQOZHEAK 7.1 Ki 3
CZWUYUYQOZHEAK 7.1 Ki 3
GGPRUUQFBUCJMT 7.1 Ki 2
WOACWYIUZSUINZ 7.1 Ki 2
DNVMLFGJFSQQDE 7.1 IC50 9
BYKPIBZUEKZONO 7.1 Ki 2
ALGQHHHCUISTSF 7.1 Ki 5
DTWANULJDRVTFI 7.1 IC50 5
MDQRTKPORXDJTI 7.1 IC50 2
CFVHNYYHCCJXDK 7.1 IC50 9
PUCADISPXQCOJH 7.1 IC50 2
HGGAFEZREIVLAZ 7.1 Ki 2
HDKROIJMOQEIJT 7.0 Ki 2
UEUSVFILMLMQMI 7.0 Ki 2
YGDUPQPZKGHOEN 7.0 IC50 2
CLNHOZKBDJOIQN 7.0 Ki 2
IAIFJGLEPUYUIM 7.0 Ki 2
JXZZSCMQQYPMOI 7.0 IC50 2
MTXSIJUGVMTTMU 7.0 Ki 3
DYSCFNKIZDWMSK 7.0 Ki 2
RDTCPZXZWHKOTD 7.0 Ki 2
SGTIJQPRESNGSP 7.0 Ki 2
OREHKCAJBKZGSF 7.0 Ki 3
TVQVEBXIMQEOQV 7.0 Ki 3
ALSKYCOJJPXPFS 7.0 IC50 3
OQLGGCKCIDDCBN 7.0 IC50 2
2D structure