Target Details
UniProt ACP43681
Gene SymbolCHRNA4
Protein NameNeuronal acetylcholine receptor subunit alpha-4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 755
  • Clinical molecules 0
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (755)
InChIKey pChEMBL Type Targets Clinical
JQSHBVHOMNKWFT 7.5 Ki 6
MVICTLGKGURDRL 7.5 Ki 2
UXOBDWKUWQKDRV 7.5 Ki 2
UYZAXUWVJGHEFL 7.5 IC50 3
GJGPBQPYTQJXLG 7.5 Ki 2
ONDDMIQCYQALKD 7.5 Ki 2
PKAUAOBCDVMNHY 7.5 Ki 2
SUAOTTUOTKDAFW 7.5 Ki 2
FUTCURITYYGPTL 7.5 Ki 2
HKLZABNBARUZMN 7.5 Ki 2
SYMAJWVHHBJSJV 7.5 IC50 8
VGHRMGBKIWAGMS 7.5 Ki 2
ALGQHHHCUISTSF 7.5 Ki 3
LHDBWAIRCLWNKW 7.5 Ki 2
AKHCKCPDLAYHDW 7.4 IC50 4
ALGQHHHCUISTSF 7.4 Ki 5
DDDMGCMKOCLAAT 7.4 IC50 8
NEWJHZNVOKNDPN 7.4 Ki 2
SUPRUPHAEXPGPF 7.4 Ki 2
DGQVZUDAKWRJPY 7.4 IC50 8
XEGIBXIZNONLNZ 7.4 Ki 2
JVTWFZWFTGAAGI 7.4 Ki 2
PYSCVJMLJRHJGJ 7.4 Ki 2
YLTIOICAHCAKID 7.4 Ki 2
NLQQWPDBPOHVHB 7.4 Ki 2
VFQWXRPPTRICFE 7.4 Ki 2
SFSMPEDWDOLQDX 7.4 IC50 2
SOEBPVQMXRKIOZ 7.4 IC50 4
XCORZZYKCQYSQJ 7.4 Ki 2
ZZWUEOYQVWAKCJ 7.4 IC50 9
BRRKZDRFDMYVGP 7.4 Ki 2
HFIMLFRJUJSWHZ 7.4 Ki 2
AZKMTKVSVYHHAA 7.4 IC50 4
IWPPBJFNTXUNGJ 7.4 Ki 2
ORHMDEPRGDBBCN 7.4 Ki 2
PXVQMUATEFMGFD 7.4 IC50 2
JRPWUGPYWRJACU 7.3 IC50 8
KPCBJGYPNGGQFN 7.3 Ki 2
NZWMSQXPQAEDAS 7.3 Ki 4
PNTLWGGPNDUEGL 7.3 Ki 2
TYCKRCIGLWSVCK 7.3 Ki 2
AZKMTKVSVYHHAA 7.3 IC50 4
CSIAFHYCIBJKSC 7.3 IC50 2
BDIVMECULLJBMU 7.3 Ki 2
DQLLEORXWPVYGE 7.3 IC50 2
KZXHYOKRCVIUQQ 7.3 IC50 2
NMIIKXFGCKOYRV 7.3 IC50 2
NZGNBOYHACXVNU 7.3 Ki 3
RBLSIFSCIAMBSU 7.3 IC50 2
YOGAMLRQMJSVCJ 7.3 Ki 2
2D structure