Target Details
| UniProt AC | P43490 |
|---|---|
| Gene Symbol | NAMPT |
| Protein Name | Nicotinamide phosphoribosyltransferase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18127 (NAMPT_N) PF04095 (NAPRTase) |
Summary
- Multi-target molecules 146
- Clinical molecules 0
- Avg pChEMBL 7.34
KEGG Pathways (3)
Active Molecules (146)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SHNBLWMBWXIKMR
|
9.0 | IC50 | 2 | — | |
BOIPLTNGIAPDBY
|
8.7 | IC50 | 5 | — | |
FSKWZBIVMXYVIB
|
8.7 | IC50 | 2 | — | |
ORDWPEHFKJXJKD
|
8.5 | IC50 | 2 | — | |
KPBNHDGDUADAGP
|
8.5 | IC50 | 2 | — | |
SJMQTTISZPIKBR
|
8.5 | IC50 | 2 | — | |
YERMBKYNILMCNC
|
8.4 | IC50 | 3 | — | |
ZZZBYLFRFPPGEA
|
8.4 | IC50 | 2 | — | |
GCNBJSNHYPKHIT
|
8.4 | IC50 | 3 | — | |
MOQYJMVBPKWDGC
|
8.3 | IC50 | 3 | — | |
XRDVXQQZLHVEQZ
|
8.3 | IC50 | 2 | — | |
CBGMGQVEMRTNGL
|
8.3 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
8.3 | Kd | 1075 | — | |
LKBHAGGICJWHQQ
|
8.2 | IC50 | 2 | — | |
JPTLLIYJDQIUGS
|
8.2 | IC50 | 2 | — | |
BRXRBZMRJJFGCH
|
8.2 | IC50 | 2 | — | |
XYGJYMRXHGHGNB
|
8.2 | IC50 | 2 | — | |
CBGMGQVEMRTNGL
|
8.1 | IC50 | 3 | — | |
DZFCBWGZQNGTQH
|
8.1 | IC50 | 2 | — | |
GUOKRDAMSCOAIA
|
8.1 | IC50 | 2 | — | |
YKTUZLHYXSJRBO
|
8.1 | IC50 | 2 | — | |
DPYKXHOJAOLOOC
|
8.1 | IC50 | 2 | — | |
OBYJQKZNRUOYGF
|
8.0 | IC50 | 2 | — | |
IFEXCZMSTXWJSK
|
8.0 | IC50 | 3 | — | |
AUXWZPVOQCZHSP
|
8.0 | IC50 | 2 | — | |
BGNOECVQVUFFHE
|
8.0 | IC50 | 2 | — | |
GCBARIQAGXVYET
|
8.0 | IC50 | 2 | — | |
AXOSMMGWCJFHKI
|
8.0 | IC50 | 2 | — | |
BIFUICSRZIQHFK
|
8.0 | IC50 | 2 | — | |
QBTMLSOSPORBBU
|
8.0 | IC50 | 2 | — | |
KBESGXIOIAXYIG
|
7.9 | IC50 | 2 | — | |
MIKRIGQVWBXZCR
|
7.9 | IC50 | 2 | — | |
QODUOXJBXDHDHN
|
7.9 | IC50 | 2 | — | |
CFPQKOXDIQRGKQ
|
7.9 | IC50 | 2 | — | |
SYEBAIPAXRFBFO
|
7.9 | IC50 | 2 | — | |
USNBTXLPADLVFT
|
7.9 | IC50 | 2 | — | |
BGECQVFGWHCTBJ
|
7.8 | IC50 | 2 | — | |
MINLAVWRIIAIGN
|
7.8 | IC50 | 2 | — | |
ROEPGCSNAWAJRM
|
7.8 | IC50 | 2 | — | |
HKRNGLFQUVCSOL
|
7.8 | IC50 | 2 | — | |
IPFCGFBLRONVPM
|
7.8 | IC50 | 2 | — | |
RBVSKBDEAXWXGR
|
7.8 | IC50 | 7 | — | |
VGOAFCLCBYDTTL
|
7.8 | IC50 | 2 | — | |
NMNMXZAMLXAEMU
|
7.8 | IC50 | 2 | — | |
DQXRTBMMUDAJNA
|
7.7 | IC50 | 2 | — | |
FVLQFSUNDROJBC
|
7.7 | IC50 | 2 | — | |
HVZNSUOYEMWTPR
|
7.7 | IC50 | 2 | — | |
WSTLKKSKCYMNAA
|
7.7 | IC50 | 7 | — | |
OMXUTMOTZCFLDJ
|
7.7 | IC50 | 2 | — | |
GBWFXYVAVDSWDW
|
7.7 | IC50 | 2 | — |