Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MHROCFGPXVNJFS
|
7.3 | IC50 | 3 | — | |
VPFQXVNSENBLHV
|
7.3 | IC50 | 4 | — | |
IUVDZGOUQXJDQC
|
7.2 | IC50 | 2 | Yes | |
JSARQMZOESQGPT
|
7.2 | IC50 | 3 | — | |
RCXLHSLQXPURIJ
|
7.2 | IC50 | 2 | — | |
XFIFRGSEYNEXIW
|
7.2 | IC50 | 2 | — | |
CTKOGVDXPJXWDZ
|
7.2 | IC50 | 2 | — | |
FEUBLBMLMVBROW
|
7.2 | IC50 | 2 | — | |
KKBSRZBNVASLTJ
|
7.2 | IC50 | 3 | — | |
ODPFOHRTWMCIJT
|
7.2 | IC50 | 3 | — | |
PCEDTTMLXHLGED
|
7.2 | IC50 | 2 | — | |
RPHZNUQELARGGG
|
7.2 | IC50 | 3 | — | |
SUCOEVXSLGWMLL
|
7.2 | IC50 | 3 | — | |
VGQAOTJFWQGYRB
|
7.2 | IC50 | 2 | — | |
QVZIZZNXCLSQQR
|
7.2 | IC50 | 3 | — | |
SUOCOHZLBGRVQJ
|
7.2 | IC50 | 2 | — | |
VWGMFKBQYRNIIN
|
7.2 | IC50 | 3 | — | |
LZAOAQYGUGHFQO
|
7.2 | IC50 | 4 | — | |
VSQDAQJVIALSGZ
|
7.2 | IC50 | 3 | — | |
AJOLXGKMRXNPKQ
|
7.2 | IC50 | 4 | — | |
CJRXFUKGUWDQNO
|
7.2 | IC50 | 3 | — | |
JDAQJEHWJCXAFI
|
7.2 | IC50 | 4 | — | |
VWGMFKBQYRNIIN
|
7.2 | IC50 | 3 | — | |
WDZOSPABBUJVMV
|
7.2 | IC50 | 3 | — | |
AIQDZMUPVYDVLB
|
7.2 | Ki | 48 | — | |
BIKYDWLMTPRSQL
|
7.2 | Ki | 50 | — | |
CPQXTCRENIMNFB
|
7.2 | IC50 | 2 | — | |
DGJNSNHNZJVEFO
|
7.2 | IC50 | 3 | — | |
GPYGSYSPXHEXTJ
|
7.2 | IC50 | 3 | — | |
KFXHPWUOUVDXSQ
|
7.2 | IC50 | 3 | — | |
KRIUNPBAQZGFQA
|
7.2 | Ki | 76 | — | |
KVPNQKXHQVOBDL
|
7.2 | IC50 | 2 | — | |
LYNBNVBMAGDJRW
|
7.2 | Ki | 81 | — | |
NTTIWAXCPUSMSY
|
7.2 | IC50 | 3 | — | |
YFVHXPJXPIIXGA
|
7.2 | IC50 | 2 | — | |
BSTCRUFJLBKYMG
|
7.2 | IC50 | 4 | — | |
GENGRGPVHLFFDS
|
7.2 | IC50 | 3 | — | |
NZEUGQYGRHEHEG
|
7.2 | IC50 | 3 | — | |
ZZSBPGIGIUFJRA
|
7.2 | Kd | 46 | — | |
CXXHIMHTNIDPAR
|
7.2 | IC50 | 3 | Yes | |
GVWNNKNAVOPJNV
|
7.2 | IC50 | 2 | — | |
VAUWNNIXFMIEBF
|
7.2 | IC50 | 3 | — | |
LZQTVVQZQUWSAI
|
7.2 | IC50 | 4 | Yes | |
RQRUNCDCHJDCDE
|
7.2 | IC50 | 3 | — | |
VSXCXKDGHBAKDZ
|
7.2 | IC50 | 3 | — | |
ZOJJTNITQOBIGV
|
7.2 | IC50 | 3 | — | |
CLKZDZYGBHNPSM
|
7.2 | IC50 | 2 | — | |
QSSIMBOFXQKHMK
|
7.2 | IC50 | 2 | — | |
AFMLPWWCVUSWHH
|
7.1 | IC50 | 3 | — | |
AUTVJIYXOFOONY
|
7.1 | IC50 | 2 | — |