Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JATDSOCHDDNIMP
|
7.4 | IC50 | 3 | — | |
WCSCGZHKZNEMNJ
|
7.4 | IC50 | 4 | — | |
GIJURJWFWCGLHN
|
7.4 | IC50 | 2 | — | |
HJCJFGMPMNBXRW
|
7.4 | IC50 | 2 | — | |
BANXPZGDYGVXOC
|
7.4 | IC50 | 4 | — | |
PTMVPXQFPYJIMN
|
7.4 | IC50 | 4 | — | |
UMXBELQMJUPJRY
|
7.4 | IC50 | 3 | — | |
VFRGUPCPOYDATL
|
7.4 | IC50 | 3 | — | |
HZKOUKPIDXDOOI
|
7.4 | IC50 | 4 | — | |
KDRIQANXEFIHCL
|
7.4 | IC50 | 4 | — | |
YEHCNYAQEBQCCS
|
7.4 | Ki | 74 | — | |
FQNFLNSVHWCZML
|
7.4 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.4 | IC50 | 220 | — | |
OSVUGUHRKMMBSE
|
7.4 | Kd | 170 | — | |
YSFGCARYACLFDS
|
7.4 | Ki | 7 | Yes | |
AVUUHIYJPTWYNX
|
7.4 | IC50 | 9 | — | |
CZNVSHUEQYXNKX
|
7.4 | IC50 | 3 | — | |
HUMIGOFJWQKXPY
|
7.4 | IC50 | 3 | — | |
LYADGAGFYYXXIO
|
7.4 | IC50 | 82 | — | |
NZIYWLJVQWAPEO
|
7.4 | IC50 | 2 | — | |
VLRRDESRPRRNAD
|
7.4 | IC50 | 4 | — | |
YNSRIXGBOYZSBO
|
7.4 | IC50 | 3 | — | |
BJJRLHLFUBMTBH
|
7.4 | IC50 | 3 | — | |
DCAMTYGKRNMTNB
|
7.4 | IC50 | 2 | — | |
GEATXDJAPAHPTP
|
7.4 | IC50 | 10 | — | |
PSKCCPWOWLPVFR
|
7.3 | IC50 | 3 | — | |
ZTMATBOBWAXBCV
|
7.3 | IC50 | 4 | — | |
ZZUSFIPRLCGKQL
|
7.3 | IC50 | 4 | — | |
BJALGJWVBDCWDU
|
7.3 | IC50 | 2 | — | |
KVBBSBPIPKLJCO
|
7.3 | IC50 | 3 | — | |
PAZVWIGCRYUCKP
|
7.3 | IC50 | 4 | — | |
XDWGWOIJGUXMSS
|
7.3 | IC50 | 2 | — | |
FOVSNASTDPXXSC
|
7.3 | IC50 | 2 | — | |
JOUPQTNCMDHNRF
|
7.3 | IC50 | 4 | — | |
VKBFHTIUXUCYRQ
|
7.3 | Ki | 66 | — | |
WBLZAYYLYJCMTJ
|
7.3 | IC50 | 3 | — | |
WPHKIQPVPYJNAX
|
7.3 | Ki | 81 | — | |
ZKLJKKASNXVQBZ
|
7.3 | Ki | 27 | — | |
CYKJKKJPMBDBAT
|
7.3 | IC50 | 4 | — | |
FPWCREKHIZDTGO
|
7.3 | IC50 | 3 | — | |
JSEJMGKNQGRPEI
|
7.3 | IC50 | 3 | — | |
VFQNGIVBLUWECA
|
7.3 | IC50 | 4 | — | |
ZBQANXLXZIWFJV
|
7.3 | IC50 | 3 | — | |
DHSZWTFDQUUKJT
|
7.3 | IC50 | 3 | — | |
URWLZYRKQMJGBE
|
7.3 | IC50 | 2 | — | |
UUGFFVXOVKEYMH
|
7.3 | IC50 | 2 | — | |
BVUUQTZSOCAXST
|
7.3 | IC50 | 3 | — | |
NSVUVPGLZGFORM
|
7.3 | IC50 | 3 | — | |
PEDMIJDFAWDUDE
|
7.3 | IC50 | 3 | — | |
KAXFCXIHQXDECG
|
7.3 | IC50 | 4 | — |