Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RYZDJZFSIODRQX
|
7.5 | IC50 | 2 | — | |
SFVSAJFMIQDDRE
|
7.5 | IC50 | 2 | — | |
SLWNSBACHGTCSL
|
7.5 | IC50 | 2 | — | |
STUXZVYNMDRZHE
|
7.5 | IC50 | 2 | — | |
SYEPZUJMAPZEEN
|
7.5 | IC50 | 2 | — | |
UJFNGXNNRFLOJF
|
7.5 | IC50 | 2 | — | |
UYPKOPXCRRSNHM
|
7.5 | IC50 | 2 | — | |
VOYFDZFWQMVMTM
|
7.5 | IC50 | 2 | — | |
WBBZJXHOJATBAX
|
7.5 | IC50 | 4 | — | |
WSMPCKSTTVSVQF
|
7.5 | IC50 | 2 | — | |
WTBBLBQFQMOQBJ
|
7.5 | IC50 | 2 | — | |
XZHMSXGDMVVRPD
|
7.5 | IC50 | 2 | — | |
XZXUMBFQVUKVQC
|
7.5 | IC50 | 2 | — | |
YBHNNEQRDMHSQQ
|
7.5 | IC50 | 2 | — | |
YKKVLDDNAYHXNZ
|
7.5 | IC50 | 2 | — | |
YNBDBXIEAYCZCT
|
7.5 | IC50 | 2 | — | |
ZLKXZPXDOZIMOT
|
7.5 | IC50 | 2 | — | |
ZXQCYVYVYRCBNM
|
7.5 | IC50 | 2 | — | |
ZZDMLBASKXCHAM
|
7.5 | IC50 | 2 | — | |
TZUDPPUGEPGOHM
|
7.5 | IC50 | 2 | — | |
WIAJWJSFVQRBAD
|
7.5 | IC50 | 3 | — | |
GCBJDOWIQHMCMR
|
7.5 | Ki | 84 | — | |
GQUIEPYFROOKLV
|
7.5 | IC50 | 3 | — | |
HSODWQGVXRNOEV
|
7.5 | IC50 | 3 | — | |
MKAHLUQCHFLGCS
|
7.5 | IC50 | 2 | — | |
RYYNGWLOYLRZLK
|
7.5 | Ki | 104 | — | |
XVVANFOECICSLK
|
7.5 | IC50 | 4 | — | |
ZLVOTRRGLSDLPF
|
7.5 | Ki | 36 | — | |
ZOBKJVAECISXJA
|
7.5 | IC50 | 2 | — | |
QIYHYLDEYCTUSQ
|
7.5 | IC50 | 2 | — | |
DNNZXXBLUGPLSI
|
7.5 | IC50 | 2 | — | |
GPPNXVDUQMDEAO
|
7.5 | IC50 | 3 | — | |
KEYJNCXZEKAAGP
|
7.5 | IC50 | 3 | — | |
XFSGWODALIPICT
|
7.5 | IC50 | 2 | — | |
YXGPQZLIIOQQAZ
|
7.5 | IC50 | 2 | — | |
ZRDDQLVMSUCMGD
|
7.5 | IC50 | 3 | — | |
CLRSATALQPIPQY
|
7.5 | IC50 | 3 | — | |
HAVMBPZPTGEWPJ
|
7.5 | IC50 | 4 | — | |
KBDMNNVCGCQHGS
|
7.5 | IC50 | 3 | — | |
LKZAFVLIMSKDQX
|
7.5 | IC50 | 3 | — | |
BEMAXRGCROABFF
|
7.5 | IC50 | 4 | — | |
DMZBGGYSGOPZET
|
7.5 | IC50 | 4 | — | |
FPQNRXITKTZFMF
|
7.5 | IC50 | 13 | — | |
JBBNRIFQSNWZOK
|
7.5 | IC50 | 4 | — | |
OSOIKRIQGXULMU
|
7.5 | IC50 | 3 | — | |
XEJOYWXISYDXMO
|
7.5 | IC50 | 2 | — | |
HMMIVTXSLFBBHC
|
7.4 | IC50 | 4 | — | |
KBPYMFSSFLOJPH
|
7.4 | IC50 | 4 | — | |
NJIAKNWTIVDSDA
|
7.4 | IC50 | 2 | — | |
WWSVFJIFHQKQLY
|
7.4 | IC50 | 3 | — |