Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AMUSCCPWKQVJSJ
|
7.5 | IC50 | 4 | — | |
IEUYALOEFWZLQN
|
7.5 | IC50 | 4 | — | |
AJXVRZSFKIWMPE
|
7.5 | IC50 | 2 | — | |
BDJHLYKXLGPKMN
|
7.5 | IC50 | 2 | — | |
BGYRXGQWAZXEDS
|
7.5 | IC50 | 2 | — | |
BJFPPTIKXSPLBJ
|
7.5 | IC50 | 2 | — | |
BQXZIESXWIBBFW
|
7.5 | IC50 | 2 | — | |
BTCNCQSGGFCVFV
|
7.5 | IC50 | 2 | — | |
BVIZVFPBEYCYPX
|
7.5 | IC50 | 2 | — | |
DCSJUPXLDMJOJR
|
7.5 | IC50 | 2 | — | |
DECWCGJHVBGDPC
|
7.5 | IC50 | 2 | — | |
FBASVZLYAFUGQZ
|
7.5 | IC50 | 2 | — | |
FRTDJFPREPWBPC
|
7.5 | IC50 | 2 | — | |
FZPPZFAJTHHYCH
|
7.5 | IC50 | 2 | — | |
GCVWGHNHKGVKKH
|
7.5 | IC50 | 2 | — | |
GFKWHZAGPDLSPU
|
7.5 | IC50 | 2 | — | |
GKDRMWXFWHEQQT
|
7.5 | IC50 | 7 | — | |
GNOPSCBEOSUMGK
|
7.5 | IC50 | 2 | — | |
GPMVYVKVZNUFQF
|
7.5 | IC50 | 2 | — | |
GQUBBCXAGYGOOD
|
7.5 | IC50 | 2 | — | |
GZBOYSRYJPNTCW
|
7.5 | IC50 | 2 | — | |
HEPZYOJLBLEMSQ
|
7.5 | IC50 | 2 | — | |
JLVJXSSGBIIFAL
|
7.5 | IC50 | 2 | — | |
JTFKYCKWTYYQAI
|
7.5 | IC50 | 2 | — | |
JWVJDZUFDKNXPY
|
7.5 | IC50 | 2 | — | |
JZKZBBWPVCRECL
|
7.5 | IC50 | 2 | — | |
KAZVWDLCKKDSPA
|
7.5 | IC50 | 2 | — | |
KBTZBNSTRFVKHX
|
7.5 | IC50 | 2 | — | |
KQSYWWGVMIWNOM
|
7.5 | IC50 | 3 | — | |
KTPXXXTUVSXPIH
|
7.5 | IC50 | 2 | — | |
KWQYOKQSJYMUAF
|
7.5 | IC50 | 2 | — | |
LFWPPUMWYUVLEU
|
7.5 | IC50 | 2 | — | |
LGYDROLDDQMUTM
|
7.5 | IC50 | 2 | — | |
LHSAEXHLZCPBIR
|
7.5 | IC50 | 2 | — | |
LQQOXQAYDYXSRD
|
7.5 | IC50 | 2 | — | |
MESFFTSCLYFQNJ
|
7.5 | IC50 | 2 | — | |
NLNRWZCZHGQCCE
|
7.5 | IC50 | 2 | — | |
NSXLMTSVPFZQNQ
|
7.5 | IC50 | 2 | — | |
NWQABPSTQALIAV
|
7.5 | IC50 | 2 | — | |
NXPMVEXTFYJLLS
|
7.5 | IC50 | 2 | — | |
OAKFEOPDFIPHNK
|
7.5 | IC50 | 2 | — | |
ODNKDIDXPUIXMO
|
7.5 | IC50 | 2 | — | |
OLKIASCWWMGXBI
|
7.5 | IC50 | 2 | — | |
OLPXPDAVZACRFD
|
7.5 | IC50 | 2 | — | |
OORIUXBKXNWQCU
|
7.5 | IC50 | 2 | — | |
OTAFQFUDRGUFGC
|
7.5 | IC50 | 2 | — | |
OWWGJGUSHNSKLR
|
7.5 | IC50 | 2 | — | |
QXWLCWKPJNSRRJ
|
7.5 | IC50 | 3 | — | |
RIHAPCPVSFCDSQ
|
7.5 | IC50 | 2 | — | |
RLZOYEVZHFYMTI
|
7.5 | IC50 | 2 | — |