Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SBGMPUIVPOGTGN
|
7.7 | IC50 | 4 | — | |
DMFLXIRKHPTWEU
|
7.7 | IC50 | 3 | — | |
KHGPYYFCIAISBU
|
7.7 | Ki | 31 | — | |
KJNNTUJLAMNBPE
|
7.7 | IC50 | 2 | — | |
MDMCYZGIXLRATE
|
7.7 | IC50 | 4 | — | |
MKAHLUQCHFLGCS
|
7.7 | IC50 | 2 | — | |
RCPBXCJRKDXEGJ
|
7.7 | IC50 | 4 | — | |
RHCMQQAUBJPPPW
|
7.7 | IC50 | 4 | — | |
URPHWXWGWHZRLT
|
7.7 | IC50 | 3 | — | |
ZGZVRPRSFXRGCF
|
7.7 | Ki | 76 | — | |
LGACHOLIGNCDSQ
|
7.7 | IC50 | 4 | — | |
LCMVLFWIBUQNAX
|
7.7 | IC50 | 2 | — | |
NALGZACUGTTXDW
|
7.7 | IC50 | 3 | — | |
OJKGJLKJOICLKA
|
7.7 | IC50 | 4 | — | |
YTFOAGDDMAAOPC
|
7.7 | IC50 | 3 | — | |
FDZBZSBLRVVIGJ
|
7.7 | IC50 | 2 | — | |
UPRPVDAEXQKBSI
|
7.7 | IC50 | 3 | Yes | |
CSZJFFGJPPIFRZ
|
7.6 | IC50 | 2 | — | |
KPYJFGGKRGRARF
|
7.6 | IC50 | 3 | — | |
VFCRJQKABYQLDB
|
7.6 | IC50 | 3 | — | |
AOEVEOHCGZVHSB
|
7.6 | IC50 | 3 | — | |
ARVCFDUHKZCQJL
|
7.6 | IC50 | 3 | — | |
DVZWNAWWJTZZNH
|
7.6 | IC50 | 3 | — | |
OFTHCDFOVLVBTL
|
7.6 | IC50 | 3 | — | |
VIFMVQBVAVNATG
|
7.6 | IC50 | 4 | — | |
ODRSUVBAJITCIK
|
7.6 | IC50 | 2 | — | |
WEACIVJSLZZZLC
|
7.6 | IC50 | 3 | — | |
YIQDCOAZVWPXQA
|
7.6 | IC50 | 4 | — | |
ZCWXCBKGPJOAFQ
|
7.6 | IC50 | 13 | — | |
OHFRZOITYIPIHR
|
7.6 | IC50 | 2 | — | |
XXSPPIWQGKTKEQ
|
7.6 | IC50 | 3 | — | |
DSQCTESAPJCINY
|
7.6 | IC50 | 3 | — | |
IUEXHNTZDWOAIZ
|
7.6 | IC50 | 3 | Yes | |
NXSJMRCTGYTSTK
|
7.6 | Kd | 200 | — | |
RQVLOUXWVWPIMN
|
7.6 | IC50 | 3 | — | |
SFCBIFOAGRZJNX
|
7.6 | IC50 | 22 | — | |
UNGHXZVJQQABCA
|
7.6 | IC50 | 3 | — | |
WXUNFLPVNBQMNX
|
7.6 | IC50 | 3 | — | |
YARHUYMJLJCURZ
|
7.6 | IC50 | 3 | — | |
ZEQMOMFMWDAHFG
|
7.6 | IC50 | 3 | — | |
BDZSQIOBXDJLKM
|
7.6 | IC50 | 3 | — | |
QMMSRYDOEGIITQ
|
7.6 | IC50 | 3 | — | |
VGHUYLNQBPEVLC
|
7.6 | IC50 | 2 | — | |
YVVSDMPVUOIAOS
|
7.6 | IC50 | 3 | — | |
HLVQIKPORSSRAI
|
7.6 | IC50 | 3 | — | |
CGELEDQBCPRRSA
|
7.5 | IC50 | 3 | — | |
OHTDBFPGRCKSTH
|
7.5 | IC50 | 2 | — | |
UCDYGVBDFHZXEE
|
7.5 | IC50 | 2 | — | |
VGYKFYWQDGVSRW
|
7.5 | IC50 | 3 | — | |
WAIFVHBFMAMLSV
|
7.5 | IC50 | 3 | — |