Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNGNGIHVGNTTHO
|
8.2 | IC50 | 3 | — | |
WRKCCXCCDUYPLU
|
8.2 | IC50 | 3 | — | |
WVYPOHDPGYBAGO
|
8.2 | IC50 | 4 | — | |
YCWQIUKZOZXDEM
|
8.2 | IC50 | 3 | — | |
WHVKZJNMFJXSSJ
|
8.1 | IC50 | 2 | — | |
JWQOJVOKBAAAAR
|
8.1 | Ki | 29 | — | |
AFFDEZDCXSAKBU
|
8.1 | IC50 | 4 | — | |
ALNFKLJYTICTCF
|
8.1 | IC50 | 4 | — | |
DTFJTXRGYIXMMS
|
8.1 | IC50 | 5 | — | |
IGRYEDIMNMEBBU
|
8.1 | IC50 | 9 | — | |
JEHBCDCKKVKVGB
|
8.1 | IC50 | 3 | — | |
LJMCZWSDLQFAMA
|
8.1 | IC50 | 2 | — | |
MFPLYINPSNJRRI
|
8.1 | IC50 | 3 | — | |
OKERWTBOFAFQQV
|
8.1 | IC50 | 3 | — | |
UJXIKUVGGQECLJ
|
8.1 | IC50 | 2 | — | |
URNGXAVMGITILR
|
8.1 | IC50 | 4 | — | |
YGZKTIVAVURWEZ
|
8.1 | IC50 | 3 | — | |
YWBUMBUFDDSLCR
|
8.1 | IC50 | 4 | — | |
IMHCVVDKOFKZKX
|
8.1 | IC50 | 3 | — | |
JMJSTGZRLYHCCI
|
8.1 | IC50 | 5 | — | |
MKJKFFODUSDVSK
|
8.1 | IC50 | 3 | — | |
MMEJLCRBNBQORJ
|
8.1 | IC50 | 3 | — | |
NAHNBJVIEWPVPP
|
8.1 | IC50 | 3 | — | |
NBGQQTFVANZDGQ
|
8.1 | IC50 | 2 | — | |
PEGXADGTBNRSGV
|
8.1 | IC50 | 2 | — | |
SALBBGQOFCZHKF
|
8.1 | IC50 | 3 | — | |
URRPWKVYUYOQBW
|
8.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
CAIDLKSVZKWPJK
|
8.0 | IC50 | 3 | — | |
CFIBXVQLBVNOHW
|
8.0 | Ki | 64 | — | |
FOOBTRPSYPGQSN
|
8.0 | IC50 | 2 | — | |
OJQQCSPYLMDJQP
|
8.0 | IC50 | 3 | — | |
RPFSNCZTTYGYDI
|
8.0 | IC50 | 3 | — | |
YMIJUBCSOKSFRU
|
8.0 | Ki | 87 | — | |
RASCHEQRJMEENP
|
8.0 | IC50 | 4 | — | |
UJBJWYNPUOLFIZ
|
7.9 | IC50 | 49 | — | |
AMKRSTDSNXNZMY
|
7.9 | IC50 | 4 | — | |
HKSWAIDHHZHZTD
|
7.9 | IC50 | 6 | — | |
IYRPCWRKUVTLQK
|
7.9 | IC50 | 2 | — | |
SGVBVAOVXTWIJT
|
7.9 | IC50 | 3 | — | |
TYBHAECIGHGJDF
|
7.9 | IC50 | 2 | — | |
VXYTXSCFJZRDPK
|
7.9 | IC50 | 3 | — | |
XAJQBNVFUKELGZ
|
7.9 | IC50 | 3 | — | |
YBFJEMNJNCMXOO
|
7.9 | IC50 | 3 | — | |
CZQVOIDVDAVDFW
|
7.9 | Ki | 18 | — | |
TVUWQDLBEOZVOU
|
7.9 | Ki | 41 | — | |
XZSYGIPHRZNQNN
|
7.9 | IC50 | 2 | — | |
LHYKFLNJIXCRLM
|
7.9 | IC50 | 4 | — | |
LUNIPUNUORVVSN
|
7.9 | IC50 | 4 | — | |
QGRUEQPBBBTRPN
|
7.9 | IC50 | 4 | — |