Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LWAHLSWZFUCILT
|
7.0 | IC50 | 2 | — | |
RIGZTRRKOZWKPG
|
7.0 | IC50 | 3 | — | |
DOMOLNAWFSVTTI
|
7.0 | IC50 | 3 | — | |
NUQXZGAPRUPKSX
|
7.0 | IC50 | 3 | — | |
CGAXIQIZJUFEGU
|
7.0 | IC50 | 3 | — | |
JMZYKNIQZZGAOQ
|
7.0 | IC50 | 3 | — | |
LJRBXGZFMWMQNY
|
7.0 | IC50 | 4 | — | |
MMBUUNLZGRAVKE
|
7.0 | IC50 | 3 | — | |
OTQOZFYTAOFNOL
|
7.0 | IC50 | 3 | — | |
ZZJDIXUCHFNLLD
|
7.0 | IC50 | 3 | — | |
HMBIOLBRLKAILX
|
7.0 | IC50 | 4 | — | |
IASAFHQCFSUWMI
|
7.0 | IC50 | 3 | — | |
JTERLHICJVJIRK
|
7.0 | IC50 | 3 | — | |
JWZOKAUCSUFVAV
|
7.0 | IC50 | 3 | — | |
QHHCOZDURKDLDL
|
7.0 | IC50 | 3 | — | |
LRZYYIZFBXFSJB
|
7.0 | Ki | 69 | — | |
MDZNNHJKFFMBHO
|
7.0 | IC50 | 2 | — | |
PXDLCDJCBFEYEN
|
7.0 | IC50 | 3 | — | |
SHEWRCTXFWSZHA
|
7.0 | IC50 | 3 | — | |
UAUJVWLUSNTVTA
|
7.0 | IC50 | 6 | — | |
XRIHVFZLYWJMPM
|
7.0 | IC50 | 2 | — | |
YDOPLCNFRXOHCC
|
7.0 | Ki | 28 | — | |
HNQXGEIEMKYOPM
|
7.0 | IC50 | 4 | — | |
OFYBGNCNPOQMEB
|
7.0 | IC50 | 2 | — | |
WCTNEALHPXRJMI
|
7.0 | IC50 | 3 | — | |
WLXLHHAZRRMMDZ
|
7.0 | IC50 | 2 | — | |
ZSUZNPQSAQRXJP
|
7.0 | IC50 | 4 | — | |
IPRGOVMOQCIUFP
|
7.0 | IC50 | 2 | — | |
KDXHNAAPPFDXHV
|
7.0 | IC50 | 3 | — | |
RDUBHIVRDVFUBN
|
7.0 | IC50 | 2 | — | |
CPVAUCCEUDAMED
|
7.0 | IC50 | 4 | — | |
JERWIKUDUYPNOF
|
7.0 | IC50 | 4 | — | |
KWEVSNRXKHUTLB
|
7.0 | IC50 | 3 | — | |
MLRLVVFULIQDBS
|
7.0 | IC50 | 4 | — | |
NYGKSLDYPFTJBU
|
7.0 | IC50 | 2 | Yes | |
QVVCBWMDXHAMET
|
7.0 | IC50 | 4 | — | |
LZZSVMHMGFYOIP
|
7.0 | IC50 | 2 | — | |
BGPSGELIEAWXPK
|
7.0 | IC50 | 4 | — | |
FDZBZSBLRVVIGJ
|
7.0 | IC50 | 2 | — | |
GDSGFCHLYCVDEQ
|
7.0 | IC50 | 3 | — | |
LOLPPWBBNUVNQZ
|
6.9 | Kd | 97 | Yes | |
VMFBKDNUNVTPGE
|
6.9 | IC50 | 3 | — | |
DOSNRYDSORPWBF
|
6.9 | IC50 | 3 | — | |
JTSDIOVGQDLARE
|
6.9 | IC50 | 3 | — | |
PSPWDUMROPJEGG
|
6.9 | IC50 | 3 | — | |
SOQOHBPYOHXFDZ
|
6.9 | IC50 | 3 | — | |
UQRGYUSMBHLGKA
|
6.9 | IC50 | 3 | — | |
YOSOEKMQFOYUKT
|
6.9 | IC50 | 3 | — | |
AKUFVJURRNGOQZ
|
6.9 | IC50 | 3 | — | |
CWEBLBDEUUBLRL
|
6.9 | IC50 | 4 | — |