Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GNMGBKSHAODYOO
|
7.1 | IC50 | 2 | — | |
HOJOCUCRLQRWDR
|
7.1 | IC50 | 2 | — | |
FBLUZGYSJKUSKN
|
7.1 | IC50 | 2 | — | |
KHLWYSIDXVRLRP
|
7.1 | IC50 | 2 | — | |
NMHBMUCWVDHROC
|
7.1 | IC50 | 2 | — | |
NXZOHMBZJBFOKG
|
7.1 | IC50 | 2 | — | |
ONWQCRZBUOXITQ
|
7.1 | IC50 | 2 | — | |
PLRVOIGCBGTLTD
|
7.1 | IC50 | 2 | — | |
QKCMDGMFYDDNIU
|
7.1 | IC50 | 2 | — | |
UMUNUYQBNZSRHV
|
7.1 | IC50 | 3 | — | |
UTBOYGRCMFIHJK
|
7.1 | IC50 | 3 | — | |
VDALILMQMHXDSL
|
7.1 | IC50 | 2 | — | |
VNURAGHRVHZAKJ
|
7.1 | IC50 | 2 | — | |
VNURAGHRVHZAKJ
|
7.1 | IC50 | 2 | — | |
VZEBZVKYQRSFDD
|
7.1 | IC50 | 3 | — | |
XOXJNDPEHAKNBZ
|
7.1 | IC50 | 2 | — | |
YKMKSKQQPHLCCJ
|
7.1 | IC50 | 2 | — | |
HTMINSIGYJFGEU
|
7.1 | IC50 | 3 | — | |
NTRGHFKSGIJGAD
|
7.1 | IC50 | 3 | — | |
SMTDHTZNDOVANM
|
7.1 | IC50 | 2 | — | |
UILXYBOXAAJRAE
|
7.1 | IC50 | 3 | — | |
BYMPQGHXDOZTHZ
|
7.1 | IC50 | 2 | — | |
FZMCQVGUQKFBIJ
|
7.1 | IC50 | 4 | — | |
HQXRVTFLFJNGAV
|
7.1 | IC50 | 2 | — | |
IFPPYSWJNWHOLQ
|
7.1 | Ki | 52 | Yes | |
KSBWPNWWWVOGJM
|
7.1 | IC50 | 2 | — | |
NLUPJKQOKWBWFC
|
7.1 | Ki | 69 | — | |
NZNTWOVDIXCHHS
|
7.1 | IC50 | 3 | — | |
PCQMERRARZKTPW
|
7.1 | Ki | 68 | — | |
QQWUGDVOUVUTOY
|
7.1 | Ki | 231 | Yes | |
RDNOLDWOMGZBPI
|
7.1 | IC50 | 8 | Yes | |
XHORJSJFHVABEA
|
7.1 | Ki | 49 | — | |
AEQLIHRFVYSWGR
|
7.1 | IC50 | 4 | — | |
HWLWBINIXVPIHY
|
7.1 | IC50 | 3 | — | |
DQGNRAHSEYSADB
|
7.1 | IC50 | 4 | — | |
FCHGXFUOVXKORC
|
7.1 | IC50 | 2 | — | |
IEHFKZAAIWSDQM
|
7.1 | IC50 | 3 | — | |
XLMGQVCEWMWIIG
|
7.1 | IC50 | 3 | — | |
XWCPBCVFAOFEEK
|
7.1 | IC50 | 3 | — | |
YBQBWKIOPABUPG
|
7.1 | IC50 | 2 | — | |
ZGVCPFSIDNPESN
|
7.1 | IC50 | 2 | — | |
ZNHAPHKYMMDRQX
|
7.1 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 91 | Yes | |
HJDQNNIRKWGQGL
|
7.1 | IC50 | 4 | — | |
JZLUCFJMWJDRIK
|
7.0 | IC50 | 7 | — | |
NJBJRWXJKAMYFV
|
7.0 | IC50 | 2 | — | |
NYXQIXYXIOVJPB
|
7.0 | IC50 | 2 | — | |
OXTMWMXCNQWAGP
|
7.0 | IC50 | 4 | — | |
FSRFRWLXYSIGBM
|
7.0 | IC50 | 4 | — |