Target Details
| UniProt AC | P43405 |
|---|---|
| Gene Symbol | SYK |
| Protein Name | Tyrosine-protein kinase SYK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 852
- Clinical molecules 32
- Avg pChEMBL 7.25
KEGG Pathways (17)
- B cell receptor signaling pathway
- C-type lectin receptor signaling pathway
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- Herpes simplex virus 1 infection
- Kaposi sarcoma-associated herpesvirus infection
- NF-kappa B signaling pathway
- Natural killer cell mediated cytotoxicity
- Neutrophil extracellular trap formation
- Osteoclast differentiation
- PI3K-Akt signaling pathway
- Phospholipase D signaling pathway
- Platelet activation
- Tuberculosis
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (852)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GZXRFDYECYFNCR
|
10.2 | IC50 | 2 | — | |
FNGJTJGYKVSXHA
|
10.0 | IC50 | 2 | — | |
GKSNOLIZSMVHCY
|
10.0 | IC50 | 3 | — | |
ONQXJCAIAGVKRH
|
10.0 | IC50 | 2 | — | |
QIYGHNDMIXXLHX
|
10.0 | IC50 | 2 | — | |
PZANSMJLRWEKCF
|
9.9 | IC50 | 2 | — | |
PAZNLQHSWVMGIW
|
9.7 | IC50 | 2 | — | |
DMHQDPVKKNQNCV
|
9.7 | IC50 | 3 | — | |
ISOQIZINACKWNJ
|
9.7 | IC50 | 3 | — | |
VRIPIEPFEURRFT
|
9.7 | IC50 | 2 | — | |
LSASLBFVFUJZOD
|
9.7 | IC50 | 2 | — | |
HJDDOMBYBZNDRI
|
9.6 | IC50 | 2 | — | |
IXNQUCOVJRJRGJ
|
9.5 | IC50 | 2 | — | |
WEMLZLDOVOESKB
|
9.3 | IC50 | 2 | — | |
YACNMLLIRLXUQZ
|
9.3 | IC50 | 2 | — | |
SRTUGXIMQMBQQX
|
9.2 | IC50 | 2 | — | |
HVQAATXUCFUOMV
|
9.2 | IC50 | 2 | — | |
HXCYFHWOPRZEBU
|
9.2 | IC50 | 2 | — | |
KSZAIPSQJXGBNH
|
9.1 | IC50 | 3 | — | |
MOXXQFNQDDSJHT
|
9.0 | IC50 | 6 | — | |
CUQPTMGVVQNXDH
|
9.0 | IC50 | 3 | — | |
JVEOZYRULRDCNQ
|
9.0 | IC50 | 3 | — | |
JXJVDYZUMYOTJW
|
9.0 | IC50 | 3 | — | |
OYKPWSZSBLRRPL
|
9.0 | IC50 | 11 | — | |
PVVFFEVERRIBNR
|
9.0 | IC50 | 3 | — | |
QBIUCEGPYOMVEE
|
9.0 | IC50 | 3 | — | |
SJOQLVNIVBIOCX
|
9.0 | IC50 | 2 | — | |
UTJDBKKZHLMLTN
|
9.0 | IC50 | 3 | — | |
VBAJQFDWESLMDW
|
9.0 | IC50 | 3 | — | |
XHZDAKAAKUZJHY
|
9.0 | IC50 | 4 | — | |
DTWUFJNGYFFLPH
|
8.9 | IC50 | 2 | — | |
SDBGQUQLHJSYJN
|
8.9 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.9 | IC50 | 408 | — | |
JHXAYGBXXCDEBZ
|
8.9 | IC50 | 2 | — | |
LVDAOOBTKGLDAK
|
8.9 | IC50 | 2 | — | |
TVTNEIYFFRQSMV
|
8.8 | IC50 | 2 | — | |
TXWSWFVDAJQPND
|
8.7 | IC50 | 2 | — | |
BIGXOFQDFCWJGU
|
8.7 | IC50 | 3 | — | |
CGXCGLMVTWFROO
|
8.7 | IC50 | 4 | — | |
HNASBONLOOCULQ
|
8.7 | IC50 | 2 | — | |
IRGAIDAWHGYOKD
|
8.7 | IC50 | 5 | — | |
KFJCYTXMHLMPLW
|
8.7 | IC50 | 3 | — | |
MGVWPOMQHQAMAV
|
8.7 | IC50 | 3 | — | |
PDFAYXCJHTYGHT
|
8.7 | IC50 | 2 | — | |
SATISEDUDGLGFE
|
8.7 | IC50 | 2 | — | |
XUIJEFBUBZVZFL
|
8.7 | IC50 | 4 | — | |
MJVGTLKDJSROLS
|
8.7 | IC50 | 2 | — | |
CLESKVZBGDCDJJ
|
8.5 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
8.5 | IC50 | 49 | Yes | |
IWADCUQKACLNKJ
|
8.5 | IC50 | 2 | — |