Target Details
| UniProt AC | P43403 |
|---|---|
| Gene Symbol | ZAP70 |
| Protein Name | Tyrosine-protein kinase ZAP-70 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 67
- Clinical molecules 12
- Avg pChEMBL 6.82
KEGG Pathways (9)
Associated Diseases (2)
Active Molecules (67)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GVRXIDPSFXZQGC
|
6.3 | IC50 | 4 | — | |
UPRPVDAEXQKBSI
|
6.3 | Ki | 3 | Yes | |
XAZBDQHARDGYFI
|
6.3 | IC50 | 2 | — | |
QIYHYLDEYCTUSQ
|
6.2 | Ki | 2 | — | |
ZZSBPGIGIUFJRA
|
6.2 | Kd | 46 | — | |
UCDYGVBDFHZXEE
|
6.2 | IC50 | 2 | — | |
CXXHIMHTNIDPAR
|
6.2 | Ki | 3 | Yes | |
UNGHXZVJQQABCA
|
6.2 | Ki | 3 | — | |
WTBBLBQFQMOQBJ
|
6.1 | IC50 | 2 | — | |
IUEXHNTZDWOAIZ
|
6.1 | Ki | 3 | Yes | |
LDMSFYNGFVTKRW
|
6.1 | Ki | 4 | Yes | |
KDXHNAAPPFDXHV
|
6.1 | IC50 | 3 | — | |
LZZSVMHMGFYOIP
|
6.0 | Ki | 2 | — | |
YYLKKYCXAOBSRM
|
6.0 | Kd | 191 | — | |
DMZTWOCJNVKCBW
|
6.0 | IC50 | 6 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
XOXJNDPEHAKNBZ
|
6.0 | Ki | 2 | — |