Target Details
| UniProt AC | P43403 |
|---|---|
| Gene Symbol | ZAP70 |
| Protein Name | Tyrosine-protein kinase ZAP-70 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 67
- Clinical molecules 12
- Avg pChEMBL 6.82
KEGG Pathways (9)
Associated Diseases (2)
Active Molecules (67)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GZXRFDYECYFNCR
|
8.3 | IC50 | 2 | — | |
YTOUFEQLXOWLSL
|
8.1 | IC50 | 2 | Yes | |
HKSZLNNOFSGOKW
|
8.1 | IC50 | 408 | — | |
JBBNRIFQSNWZOK
|
7.8 | IC50 | 4 | — | |
LSASLBFVFUJZOD
|
7.8 | Kd | 2 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
UILXYBOXAAJRAE
|
7.7 | IC50 | 3 | — | |
OYKPWSZSBLRRPL
|
7.6 | IC50 | 11 | — | |
NHHQJBCNYHBUSI
|
7.5 | IC50 | 220 | — | |
ZTMATBOBWAXBCV
|
7.5 | IC50 | 4 | — | |
GTMPOMUKVBZKDU
|
7.4 | IC50 | 2 | — | |
UCDYGVBDFHZXEE
|
7.4 | IC50 | 2 | — | |
LPKOEWTZGVUEJF
|
7.3 | IC50 | 3 | — | |
WCSCGZHKZNEMNJ
|
7.3 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
7.3 | IC50 | 49 | Yes | |
NQXBCUWKAWQTMT
|
7.3 | IC50 | 2 | Yes | |
LRSSMJXTQUVHEA
|
7.3 | IC50 | 2 | — | |
TXGKRVFSSHPBAJ
|
7.2 | IC50 | 11 | — | |
IXNQUCOVJRJRGJ
|
7.1 | Kd | 2 | — | |
NTTIWAXCPUSMSY
|
7.1 | IC50 | 3 | — | |
MJHOMTRKVMKCNE
|
7.1 | IC50 | 12 | — | |
LJRBXGZFMWMQNY
|
7.1 | IC50 | 4 | — | |
YISMQBFJYDFMAL
|
7.1 | IC50 | 46 | — | |
VLHKHLQNVJKAHG
|
7.0 | IC50 | 2 | — | |
UAUJVWLUSNTVTA
|
7.0 | IC50 | 6 | — | |
NXSJMRCTGYTSTK
|
7.0 | Kd | 200 | — | |
QMTFEPLRHYDWQT
|
7.0 | IC50 | 2 | — | |
JMJSTGZRLYHCCI
|
6.9 | IC50 | 5 | — | |
QQVFMNGYKNAGOD
|
6.9 | IC50 | 2 | — | |
FPQNRXITKTZFMF
|
6.9 | IC50 | 13 | — | |
QNULKTUETCUJKC
|
6.9 | IC50 | 14 | Yes | |
JZLUCFJMWJDRIK
|
6.9 | IC50 | 7 | — | |
VTOIZTHVLKSUOX
|
6.8 | IC50 | 2 | — | |
YLCFOHVAOBLAIK
|
6.7 | IC50 | 14 | — | |
BZSUCLDZAQTFQJ
|
6.7 | IC50 | 4 | — | |
DVAXQAPODFQWRX
|
6.6 | IC50 | 2 | — | |
PEGXADGTBNRSGV
|
6.6 | Ki | 2 | — | |
PFQHUUDPALIKDR
|
6.6 | IC50 | 3 | — | |
XZSYGIPHRZNQNN
|
6.6 | Ki | 2 | — | |
GQUIEPYFROOKLV
|
6.5 | Ki | 3 | — | |
RVIMFNLCTIXVKN
|
6.5 | IC50 | 4 | — | |
VPFQXVNSENBLHV
|
6.5 | IC50 | 4 | — | |
DNNZXXBLUGPLSI
|
6.5 | IC50 | 2 | — | |
LZAOAQYGUGHFQO
|
6.4 | IC50 | 4 | — | |
VSJXTUFWPAOYLC
|
6.4 | IC50 | 11 | Yes | |
BPLTVYXMXOYIBK
|
6.4 | IC50 | 9 | — | |
BPLTVYXMXOYIBK
|
6.4 | IC50 | 6 | — | |
PAZNLQHSWVMGIW
|
6.4 | Kd | 2 | — | |
LZQTVVQZQUWSAI
|
6.4 | Ki | 4 | Yes | |
GVWNNKNAVOPJNV
|
6.4 | Ki | 2 | — |