Target Details
| UniProt AC | P43250 |
|---|---|
| Gene Symbol | GRK6 |
| Protein Name | G protein-coupled receptor kinase 6 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 19
- Clinical molecules 1
- Avg pChEMBL 6.95
KEGG Pathways (3)
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ACLLLJSNOCYQOJ
|
8.1 | IC50 | 8 | — | |
GYMOXCZIQHPXOH
|
7.9 | IC50 | 6 | — | |
PTJBMQVUHYZJLN
|
7.6 | IC50 | 5 | — | |
VBNHXUAHZPDQJV
|
7.6 | IC50 | 2 | — | |
HZHXOMKYANMUKK
|
7.5 | IC50 | 2 | — | |
TWODCXKEZZLNTI
|
7.4 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.4 | IC50 | 408 | — | |
AZCHQQLGTDJHFL
|
7.1 | IC50 | 3 | — | |
NYHGUPGYNIRFGO
|
7.0 | IC50 | 2 | — | |
KFXDAXMJWYLKDE
|
7.0 | IC50 | 2 | — | |
QIKJAWWGNVSEHB
|
6.9 | IC50 | 2 | — | |
LADJEJIWLZWLBM
|
6.7 | IC50 | 2 | — | |
CNQINLDSXMBRHJ
|
6.6 | IC50 | 2 | — | |
MYVXPLSILQDDFA
|
6.6 | IC50 | 2 | — | |
XYUFCXJZFZPEJD
|
6.3 | IC50 | 23 | Yes | |
LYADGAGFYYXXIO
|
6.3 | IC50 | 82 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |