Target Details
UniProt ACP43235
Gene SymbolCTSK
Protein NameCathepsin K
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1)
Summary
  • Multi-target molecules 835
  • Clinical molecules 1
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (835)
InChIKey pChEMBL Type Targets Clinical
DAQZLXYFNHPPBP 7.7 Ki 3
HMBMWMLWZRYGBJ 7.7 Ki 2
HWJVUROICHNXPI 7.7 Ki 2
LMZYZVWKTJFLSL 7.7 Ki 2
ZSSCFBDEVDZJNE 7.7 Ki 3
DEKMUSVVANPFAA 7.7 IC50 4
DIJRHKKEXBYHGJ 7.7 Ki 2
DRRLOKQBVIVNIT 7.7 IC50 5
GIYDWKDCFUACBE 7.7 Ki 2
HADOCXLKVIUAKC 7.7 Ki 2
INQYGWSRYUSEJI 7.7 Ki 2
JJYZCBORPVSLNL 7.7 Ki 3
KSKVGJIYFXPPFQ 7.7 Ki 2
NRLBGKWSOSYHJM 7.7 IC50 4
QDIJVNXMKNMYPL 7.7 IC50 3
UIOWYXXRERXCMP 7.7 IC50 3
VQYXNZIEKJIVRK 7.7 IC50 2
VQYXNZIEKJIVRK 7.7 IC50 2
YGYPGVCFJLTCGO 7.7 Ki 3
YQKMEJDAMLDEFV 7.7 IC50 3
YKFSGPSMOHAYEG 7.7 IC50 4
ABGBBQLBNIVODC 7.7 IC50 4
KIGJQHZQBSCHKN 7.7 Ki 2
QVEPUJVWVMPMMN 7.7 Ki 2
SPFPXVZAXMQYRP 7.7 Ki 3
UZAPJVAEXMCCGK 7.7 Ki 2
WGNWEPPRWQKSKI 7.7 IC50 3
YYVYNDITYXLIBI 7.7 IC50 4
ZLXFGUGFOLETFJ 7.7 Ki 2
OFNOZMJQFVWTHP 7.7 IC50 4
AABIMOFMGWOKOP 7.7 Ki 2
APGQPPIXNOCMOK 7.7 Ki 3
FRXAKVHWABXMGZ 7.7 Ki 3
MAGUCZGWMHQBRA 7.7 Ki 2
NEJGUCSKQVFSJQ 7.7 Ki 2
NNPAUJLJTFBVRA 7.7 Ki 2
HCJPYLNVLFDHCY 7.6 IC50 3
JPQIXMPQVCDFBY 7.6 Ki 5
MANOSMRLHJERON 7.6 IC50 3
NJKWZQGOBIFPBG 7.6 IC50 3
TXNDJCXNKMIHRP 7.6 Ki 3
ZKSDUCXACMZPEQ 7.6 IC50 2
SZYYBVWPURUFRR 7.6 IC50 8
BKMARWROUWRNAF 7.6 IC50 3
GDBQQVLCIARPGH 7.6 Ki 10
RHHVUDLUXPBHLT 7.6 Ki 3
XMXQTAXOTWDYTP 7.6 IC50 3
ZBRHHBWBGUXOAL 7.6 IC50 4
ZFEZJCWWCISELK 7.6 IC50 2
MSHULPIKNRKAQH 7.6 IC50 3
2D structure