Target Details
UniProt ACP43235
Gene SymbolCTSK
Protein NameCathepsin K
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1)
Summary
  • Multi-target molecules 835
  • Clinical molecules 1
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (835)
InChIKey pChEMBL Type Targets Clinical
AEACXIXTPAQTGN 7.9 IC50 4
BSRQMYCWEZBYDT 7.9 IC50 3
LZLJBBHMBQJUSF 7.9 IC50 2
NMXQSPUYSZKXOQ 7.9 IC50 2
UACFOBWDKNMPIT 7.9 Ki 2
GPNKIBLPGGECDL 7.8 Ki 2
IDXQMTAKYJAPAU 7.8 Ki 2
LNKPBUDUCNILFJ 7.8 Ki 2
MLAYQZHQPOWWIL 7.8 IC50 3
RRUMJQWYXJECGM 7.8 Ki 2
XOEDLXYIMZDHJS 7.8 Ki 2
UHLAHTJAHQWXNZ 7.8 Ki 2
CDRBHCLTCQQBPU 7.8 IC50 2
GHDIYQHGVKVLJX 7.8 IC50 2
HCUSCRVWQSVUSO 7.8 Ki 2
NIILIYWHNBVXGZ 7.8 Ki 2
QJXVROLCYARZCT 7.8 Ki 3
UHKYDXLKAPAQBJ 7.8 Ki 3
URXJGLPDOQMDSN 7.8 Ki 2
ZAXIHIPNQZPMAW 7.8 IC50 2
CJBKRGZUEZKUHF 7.8 Ki 2
JQVMCNNSVBCHGY 7.8 Ki 2
LNAVFHDQXNMEGY 7.8 Ki 2
LRBLPKQTSFLGSX 7.8 Ki 2
MVLVSSYWLGSAFE 7.8 IC50 3
NGAUZCRIRRLFOO 7.8 IC50 2
RHJVMKIXYFKWTL 7.8 Ki 2
RQVBWCPVPXPOLA 7.8 Ki 2
VEXSUPHHAIQGGG 7.8 IC50 2
WKXBMIIFIYFZLO 7.8 Ki 3
BPWNJPXVAFVVPP 7.8 IC50 4
CRPZBEVSSSRFRT 7.8 IC50 2
GVIPJIBLWRMISS 7.8 IC50 4
HLZVKJIKNRQXFG 7.8 IC50 2
IZZLPBCQUIYOGB 7.8 IC50 4
KJSQAFPATOUENW 7.8 IC50 3
KYELOXDGOIUIAM 7.8 IC50 3
MTVNDTARQDTHDY 7.8 IC50 3
MUJGQUKMVDBOLQ 7.8 Ki 2
VVTIXYQVNYENBM 7.8 IC50 2
QNUYHZAYXDMWMT 7.8 IC50 5
WZWOSKAWLSAHCD 7.8 IC50 2
WZWOSKAWLSAHCD 7.8 IC50 2
ADBVEVDVYNSEBG 7.7 Ki 2
KCXVQPRWXYAYNA 7.7 IC50 3
LADNPCFYVROVIW 7.7 IC50 2
PHKGTCBBQTUGFZ 7.7 Ki 2
PSYFDUMOGGGSNW 7.7 Ki 2
QFROONXAYAPHSD 7.7 Ki 2
BPEQZXFPWIFQDE 7.7 Ki 2
2D structure