Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VMSZYKRQEOLBRN
|
8.1 | IC50 | 2 | — | |
VMSZYKRQEOLBRN
|
8.1 | IC50 | 2 | — | |
YYESFYZVWDKKFF
|
8.1 | Ki | 2 | — | |
AQKWFYTVDBTXNS
|
8.1 | Ki | 2 | — | |
BMFYRFFIWZYPGT
|
8.1 | IC50 | 2 | — | |
JPTCTVGEINKTLG
|
8.1 | Ki | 2 | — | |
KFZXSMATDSSFDD
|
8.1 | IC50 | 2 | — | |
MQWFPEJVMZVZBQ
|
8.1 | IC50 | 2 | — | |
OMLSDHLIAQMOAZ
|
8.1 | Ki | 2 | — | |
PQTUVUOTFUHROL
|
8.1 | IC50 | 2 | — | |
RQFQNQBNKTWWPR
|
8.1 | IC50 | 3 | — | |
UZCUBOSCRIAKSH
|
8.1 | IC50 | 3 | — | |
VJBNYTFCTIYDMG
|
8.1 | IC50 | 3 | — | |
XLBWCOXGAKGLEV
|
8.1 | Ki | 2 | — | |
GDMSYEKYXAWLNM
|
8.0 | Ki | 2 | — | |
ADOJZMMSYUTJST
|
8.0 | IC50 | 2 | — | |
DEUHRFYIQWZXMJ
|
8.0 | IC50 | 3 | — | |
FNMSKYFYFLZDOO
|
8.0 | Ki | 2 | — | |
FZHIOQHRCZUATD
|
8.0 | Ki | 2 | — | |
KKTXBHJKYUPNJF
|
8.0 | IC50 | 2 | — | |
NBYWKBORRCROGO
|
8.0 | IC50 | 2 | — | |
OKAYCQSOIKKHMZ
|
8.0 | IC50 | 3 | — | |
UDPRWQLZVHVIPZ
|
8.0 | Ki | 3 | — | |
VERRQZHHHXASLV
|
8.0 | IC50 | 2 | — | |
VERRQZHHHXASLV
|
8.0 | IC50 | 2 | — | |
YOCXNQGSQYLPLF
|
8.0 | IC50 | 2 | — | |
YTZATKBXVITBCC
|
8.0 | Ki | 2 | — | |
ZLPJZJIBBLLPIY
|
8.0 | IC50 | 3 | — | |
ZZFJAPGUVYMXSJ
|
8.0 | IC50 | 2 | — | |
MKAMNFYJFXAVNX
|
8.0 | IC50 | 3 | — | |
ADKVCJPUSODNCK
|
8.0 | IC50 | 2 | — | |
VGIWPEJPLFVKSL
|
8.0 | Ki | 4 | — | |
DNKACFADGVUWHV
|
8.0 | Ki | 2 | — | |
NZKJJBIELHRDDV
|
8.0 | Ki | 2 | — | |
OQJQSVZAPSMNLA
|
8.0 | IC50 | 2 | — | |
QZNZUAQJQNRICS
|
8.0 | Ki | 2 | — | |
UFQYUTMOGQOOFL
|
8.0 | IC50 | 2 | — | |
UJHQYDKTGZAAFX
|
8.0 | IC50 | 3 | — | |
GIQMZBQRQSROHM
|
8.0 | IC50 | 2 | — | |
RTCASLUORPXCNR
|
7.9 | IC50 | 2 | — | |
VKQOQWWJCCFELL
|
7.9 | IC50 | 4 | — | |
YTRZAWRAPFBEQT
|
7.9 | IC50 | 2 | — | |
AWEFNCACPBKWGG
|
7.9 | Ki | 3 | — | |
FJYRGAFKIGNKHD
|
7.9 | Ki | 2 | — | |
GLZGNFOBDIGKFZ
|
7.9 | IC50 | 3 | — | |
IGWMYMDMZAKLGO
|
7.9 | IC50 | 3 | — | |
OMTFVAYHUNMOKR
|
7.9 | Ki | 2 | — | |
WNBYROIOFHRCHS
|
7.9 | IC50 | 3 | — | |
WNBYROIOFHRCHS
|
7.9 | IC50 | 3 | — | |
QFRLOVNUDLMMCT
|
7.9 | IC50 | 3 | — |