Target Details
UniProt ACP43235
Gene SymbolCTSK
Protein NameCathepsin K
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1)
Summary
  • Multi-target molecules 835
  • Clinical molecules 1
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (835)
InChIKey pChEMBL Type Targets Clinical
JJLGIGBUWDYNKF 8.3 Ki 2
OIKRJCDAWZOUQV 8.3 Ki 3
ZBNVNRCRULQVAR 8.3 IC50 3
JBXZNIFMTVSEQN 8.3 IC50 4
XVXGIBWJZKQFOS 8.3 Ki 2
XVXGIBWJZKQFOS 8.3 Ki 2
DZHKQXPPMAFVCH 8.2 Ki 2
JKRUSRGXYHQECR 8.2 IC50 3
KMJURIDKPLGXEZ 8.2 Ki 2
FLDXVFAWFMLTGY 8.2 Ki 2
FNEUKBQFZSGMQF 8.2 IC50 3
JCNSDZKPNRHBPD 8.2 IC50 2
OCNRYIRRTPOMKW 8.2 IC50 3
OGODDSLNRULSMM 8.2 IC50 3
PCCGUZVUPBIHJH 8.2 IC50 2
VOWUIFRLUKZWRM 8.2 IC50 2
XCKRDANFKQJNSM 8.2 IC50 2
ZMGKSZRPSXSLQP 8.2 IC50 3
JICMCJAFBMCIIX 8.2 IC50 3
XHGOLGYGBDIOFD 8.2 IC50 3
XXWDDQJFYNJUCB 8.2 IC50 3
QPGAIIGEIAEEEV 8.2 Ki 2
RPWHXFWFWHAXEI 8.2 IC50 3
HZDRVVKBWNJMQJ 8.2 Ki 2
LIEGBEDOWUMXJS 8.2 Ki 2
LNCZYHBVFQTPDF 8.2 IC50 2
NMUUAEHBZNHTOB 8.2 Ki 2
VWGLHPDSAYQVRM 8.2 IC50 3
CZDVMEOSWMPNHD 8.1 IC50 3
QFJGHQXICGBKTL 8.1 IC50 3
SVRAIXWYUFFDBX 8.1 Ki 2
AJAZMOFONMJGNP 8.1 IC50 3
GMHBWGMFTPGDOI 8.1 IC50 3
OOESIBLDEWSAMK 8.1 IC50 2
PACZTXUZEYVPIY 8.1 IC50 2
TWOOZSOQPIWDLA 8.1 IC50 3
ZJMNNURDJNZLHH 8.1 Ki 3
AQPCFTUFFUSBNZ 8.1 IC50 2
DKJNJGMFODPLQX 8.1 IC50 2
KGQJPYFDDXZLJX 8.1 Ki 2
QFXNURNWJUSIOB 8.1 Ki 4
QUSIOUMZTUGDDD 8.1 Ki 2
SFJDJSZPQMRWML 8.1 Ki 2
XCTNQGKKNUPDFM 8.1 IC50 4
DNPXBKDRCWMFFM 8.1 Ki 2
LKVLCOTZWXWKQV 8.1 IC50 3
CQKATIOOXAEWAB 8.1 IC50 3
KIBPLHFGSWCUTN 8.1 IC50 2
QZSSZOWDSLCTPA 8.1 Ki 2
UYNKWYCAWNTQDV 8.1 Ki 3
2D structure