Target Details
UniProt ACP43235
Gene SymbolCTSK
Protein NameCathepsin K
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1)
Summary
  • Multi-target molecules 835
  • Clinical molecules 1
  • Avg pChEMBL 7.64
Top Co-occurrence Targets
Active Molecules (835)
InChIKey pChEMBL Type Targets Clinical
CABJFQPQQUDNAL 8.6 IC50 3
NSGWZYNAWLMONK 8.6 Ki 2
PCBFMIZUTVTQPF 8.6 Ki 2
UTDIUZBVSSNGOU 8.6 Ki 2
UTDIUZBVSSNGOU 8.6 Ki 2
FCAAVWUXVKZIMW 8.5 Ki 3
CDFSITIHQOZSIN 8.5 IC50 7
CXDMEJPMIGCWHH 8.5 IC50 2
HYVXUIONWPXUDB 8.5 IC50 4
INKRRADDPLEFMU 8.5 Ki 3
QGHJVLUJBRKREM 8.5 Ki 3
SNHOBOKULKSZIU 8.5 Ki 3
SZQZHZOCBPSZIO 8.5 Ki 2
UDGAMABNKKQXCJ 8.5 Ki 2
XCVJGPONRKMMGU 8.5 IC50 2
XTBBBYLRJBRVPZ 8.5 IC50 2
WZJDSWDMVYJVRT 8.5 Ki 2
CTAIZAPBSQNUAF 8.5 IC50 4
NJKBASVLBVUNMW 8.5 IC50 3
VBPPNJCVXGAZDD 8.5 IC50 5
YODJPZCMOLJXNN 8.5 Ki 4
JJNKDTWKWYLERH 8.5 IC50 3
KHXWGZGVODXABJ 8.5 Ki 4
YCGCXDDZHQMZQY 8.5 Ki 2
UEYQVOFQELMNBH 8.4 IC50 2
NHFKTEZZOWFJBK 8.4 IC50 4
BWYBBMQLUKXECQ 8.4 Ki 3
LTLYEAJONXGNFG 8.4 IC50 9
LXJSHWJYJOFWTE 8.4 Ki 4
QFKLVGHIGYFYJD 8.4 IC50 2
QQZSKYDYMQGTTF 8.4 IC50 3
RFCUHPQJTGIXFS 8.4 Ki 2
RFCUHPQJTGIXFS 8.4 Ki 2
VCOJPMHZVSQSKW 8.4 IC50 3
WOLBGFZLMWKIDO 8.4 Ki 2
XGXDWBUGQKHTSH 8.4 IC50 3
XYWJXPMKFBUDQU 8.4 Ki 2
ZOCPXKXAOXQZSF 8.4 IC50 3
MCKCVIDASJTQSU 8.3 Ki 3
VMHUZXIKHJBMFK 8.3 Ki 2
RSIVRPBUNKODPD 8.3 IC50 3
LBCGIKORTZAZTM 8.3 IC50 3
GGQXMEFMGFPZJK 8.3 Ki 2
FTYFSDKVUZSZJG 8.3 Ki 2
FXNPOQWGWLQWDM 8.3 Ki 2
IJVAYUWTLKHHKT 8.3 Ki 2
MQRWKSMRQVMZEN 8.3 IC50 4
OSUGJHDCNKZEDV 8.3 Ki 4
VYRSXJDNPISAMG 8.3 IC50 2
YUMYYTORLYHUFW 8.3 IC50 5
2D structure