Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZQXYZTRTLGOBEJ
|
9.5 | IC50 | 4 | — | |
ONABDOMWRCXLPX
|
9.5 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
9.4 | IC50 | 6 | — | |
STBKPRWJLMIORW
|
9.4 | IC50 | 2 | — | |
TVZIAMLRFHJDFH
|
9.4 | IC50 | 2 | — | |
ZDEDZSBCUXOIBZ
|
9.4 | IC50 | 2 | — | |
VMUVUIMPWWGDDN
|
9.3 | IC50 | 4 | — | |
KQYFHIPAAHRARB
|
9.3 | Ki | 4 | — | |
CIUWURDWXWNZCC
|
9.3 | IC50 | 2 | — | |
PACZTXUZEYVPIY
|
9.3 | IC50 | 3 | — | |
ZLZXUNHJWVLGTE
|
9.3 | IC50 | 4 | — | |
BSPZFJDYQHDZNR
|
9.2 | IC50 | 7 | — | |
DAJBUTDDFYLLSS
|
9.2 | IC50 | 3 | — | |
FIVYCSWOCXEWSE
|
9.2 | IC50 | 4 | — | |
LLEYFYXOCVQUBI
|
9.2 | IC50 | 6 | — | |
NFCWEXBTWZUZMD
|
9.2 | IC50 | 3 | — | |
VQKRNTTUZDCHOZ
|
9.2 | Ki | 3 | — | |
UGAZRSHSXNNYTK
|
9.2 | Ki | 5 | — | |
AQQFLUKPFDHDKF
|
9.2 | Ki | 2 | — | |
QVDJMLQSYRSZKC
|
9.1 | Ki | 6 | Yes | |
LNPHKLHXDNQJOM
|
9.1 | Ki | 2 | — | |
OXTNJKCSQHCZQO
|
9.1 | Ki | 2 | — | |
VPRPGHWVFIVNRD
|
9.1 | IC50 | 3 | — | |
IBVYZTXPOAZNHM
|
9.1 | IC50 | 3 | — | |
QTPYRNAKLBXKNP
|
9.1 | IC50 | 3 | — | |
IVHANADPEKMLMO
|
9.1 | Ki | 2 | — | |
UTUSRLWZFBUDAM
|
9.1 | Ki | 4 | — | |
HDTFLVIWSNGBAC
|
9.1 | IC50 | 3 | — | |
LFKWIZQIKIHFJP
|
9.1 | Ki | 4 | — | |
POELQXXPKHMGFF
|
9.1 | IC50 | 7 | — | |
KXZLSPLTNDGSNP
|
9.0 | IC50 | 3 | — | |
LBKFBCRXNHVDOJ
|
9.0 | IC50 | 2 | — | |
VUVLQWZOUOAKHY
|
9.0 | IC50 | 4 | — | |
VUVLQWZOUOAKHY
|
9.0 | IC50 | 4 | — | |
XRIMMJTYAWYVEL
|
9.0 | Ki | 4 | — | |
JOBQWEVUTRQKOK
|
9.0 | IC50 | 3 | — | |
NSXOUETVXVPOFT
|
9.0 | IC50 | 4 | — | |
OCAFABUKPVDIBK
|
9.0 | IC50 | 3 | — | |
OSDDWOIIKLKPAK
|
9.0 | IC50 | 2 | — | |
PBNCMMUOTWZQFN
|
9.0 | IC50 | 2 | — | |
RATKYIAPMTVTOZ
|
9.0 | Ki | 2 | — | |
VBPPTMDMNMVDMW
|
9.0 | IC50 | 2 | — | |
ZBLLHXCRPWKVCY
|
9.0 | IC50 | 3 | — | |
VPRPGHWVFIVNRD
|
9.0 | IC50 | 3 | — | |
QKEJYPYBQSRFEX
|
9.0 | IC50 | 3 | — | |
SSEVORDVTHEORU
|
9.0 | IC50 | 2 | — | |
GBMRHPFMWMDHIG
|
8.9 | IC50 | 2 | — | |
MTWFVGHXLPKAPY
|
8.9 | IC50 | 2 | — | |
YUMYYTORLYHUFW
|
8.9 | Ki | 3 | — | |
YUMYYTORLYHUFW
|
8.9 | Ki | 3 | — |