Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VUNCDQVIHHNTRK
|
6.7 | Ki | 2 | — | |
YFUZVOLEKQFVCQ
|
6.7 | IC50 | 5 | — | |
BTCWCLVJZODNRF
|
6.7 | Ki | 3 | — | |
FSIREUUIWZPQTN
|
6.7 | IC50 | 3 | — | |
ZXHXXGCJLDYHEB
|
6.7 | IC50 | 2 | — | |
BMVCVCAQOQNEAB
|
6.7 | IC50 | 2 | — | |
QHDNYLUGIIWMMG
|
6.7 | IC50 | 2 | — | |
FXILBKWGQQHVJE
|
6.7 | IC50 | 2 | — | |
KGWCBORIZBPTEG
|
6.7 | IC50 | 4 | — | |
MOUOCLJGWKHZBT
|
6.7 | IC50 | 3 | — | |
RUHJZXDUKDCUQP
|
6.7 | IC50 | 2 | — | |
SBCCNMDXOPPQRI
|
6.7 | IC50 | 2 | — | |
UHCQVUSKXCWEQL
|
6.7 | IC50 | 2 | — | |
ZFWPNYQSYFERIU
|
6.7 | IC50 | 2 | — | |
CJFRYKIQLJALCT
|
6.7 | IC50 | 4 | — | |
FDOGVSMVDMDCMI
|
6.7 | IC50 | 4 | — | |
FTEBHYTXXKJNBZ
|
6.7 | IC50 | 3 | — | |
KITWVDOAAQWOFA
|
6.7 | Ki | 2 | — | |
XMQRZKLVBVOGHY
|
6.7 | Ki | 2 | — | |
FFYFBFASQTXZRA
|
6.6 | Ki | 3 | — | |
GMUXXTCOBZDVFS
|
6.6 | Ki | 4 | — | |
JPQIXMPQVCDFBY
|
6.6 | Ki | 2 | — | |
TVUDUONIRJXXCP
|
6.6 | Ki | 4 | — | |
HTRJYWNEPLFXGA
|
6.6 | IC50 | 2 | — | |
IXULIQOVYWLEAV
|
6.6 | IC50 | 3 | — | |
LEQCOSRDVNJGQU
|
6.6 | IC50 | 2 | — | |
UAEAHQWORKLQQF
|
6.6 | Ki | 2 | — | |
HMWRNUSDQUTLEW
|
6.6 | Ki | 2 | — | |
AQSMXTCYTUNCFB
|
6.6 | IC50 | 3 | — | |
GUBCDSPWYILVJH
|
6.6 | IC50 | 4 | — | |
MISDWDKRXRRBHF
|
6.6 | Ki | 3 | — | |
ORFRHRXPOJVPSF
|
6.6 | IC50 | 2 | — | |
OWXGOHWYUAIZNU
|
6.6 | IC50 | 2 | — | |
ARKFDHGHDFNOKH
|
6.6 | Ki | 4 | — | |
DCDFVKDUIGKXRF
|
6.6 | Ki | 2 | — | |
HYOBEPVMGGOORB
|
6.6 | Ki | 2 | — | |
POPLFVJHDAWIDM
|
6.6 | IC50 | 3 | — | |
QXQAFIAKTXDYFI
|
6.6 | Ki | 3 | — | |
BKFPUUQAFFNOOU
|
6.6 | IC50 | 2 | — | |
BTHLZKFLHOUZNZ
|
6.6 | Ki | 2 | — | |
SEBANXBXZIIACF
|
6.6 | IC50 | 3 | — | |
WHGKLAHPYJXNIO
|
6.6 | Ki | 2 | — | |
NBJUMGLMSOHJOR
|
6.5 | IC50 | 2 | — | |
OWIUZHNSDNFERG
|
6.5 | IC50 | 2 | — | |
QHQDWAPRBHWGKK
|
6.5 | IC50 | 2 | — | |
CCMLFCPHJPWXFB
|
6.5 | IC50 | 3 | — | |
GLDNCRGNTMYXND
|
6.5 | IC50 | 3 | — | |
LJJZYTHITLGKFY
|
6.5 | IC50 | 2 | — | |
YOJBVDOLDVVFSO
|
6.5 | Ki | 2 | — | |
BBECUGKQKLZBOE
|
6.5 | Ki | 4 | — |