Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBALKZAVEMIILY
|
6.9 | IC50 | 4 | — | |
NJIHVNVGSAOPKR
|
6.9 | Ki | 2 | — | |
OLIMBXKACVCIMM
|
6.9 | IC50 | 3 | — | |
UHFLVCRUHSLCAK
|
6.9 | IC50 | 2 | — | |
GAVRQMDMBSIEDN
|
6.9 | IC50 | 2 | — | |
GLJZTHKUTGOBFU
|
6.9 | Ki | 4 | — | |
LDQAOERTIHJZOI
|
6.9 | Ki | 2 | — | |
OMQSGXGRANQGLE
|
6.9 | Ki | 2 | — | |
YCPWFRMYSJKIIG
|
6.9 | IC50 | 4 | — | |
ACGFKLACOBPYKQ
|
6.9 | IC50 | 4 | — | |
ACGFKLACOBPYKQ
|
6.9 | IC50 | 4 | — | |
GXDULIFEODNFQZ
|
6.9 | IC50 | 4 | — | |
GXDULIFEODNFQZ
|
6.9 | IC50 | 4 | — | |
TXEWBLHLNYNUAG
|
6.9 | IC50 | 4 | — | |
TXEWBLHLNYNUAG
|
6.9 | IC50 | 4 | — | |
YEOKXFGVPJIODJ
|
6.9 | IC50 | 2 | — | |
LSACLAVWRMJGMI
|
6.9 | Ki | 2 | — | |
WYBFWCUCYMPPNV
|
6.9 | IC50 | 3 | — | |
HCLPDRDQDGUFSD
|
6.9 | IC50 | 4 | — | |
XGEOFLZCNAEENF
|
6.9 | Ki | 3 | — | |
CRBJCNGWYFLJPW
|
6.8 | IC50 | 4 | — | |
GGNPRFIUKYTFLP
|
6.8 | Ki | 2 | — | |
JIGGOBDMVDMNHC
|
6.8 | IC50 | 2 | — | |
NBEARLDWGIZSTM
|
6.8 | IC50 | 3 | — | |
SLQWQWLTTFJRHB
|
6.8 | IC50 | 2 | — | |
OKUSXRJDJJJKGN
|
6.8 | IC50 | 2 | — | |
WWVOULFEIOXZLF
|
6.8 | IC50 | 4 | — | |
UXVCQUAZYFJMPX
|
6.8 | IC50 | 2 | — | |
HDQBKIWKLLGTGO
|
6.8 | IC50 | 4 | — | |
QTCAQPIWOIDXIR
|
6.8 | Ki | 2 | — | |
QURFFOZMRDDRRV
|
6.8 | Ki | 3 | — | |
UKNHAMBXKRGPNU
|
6.8 | Ki | 2 | — | |
YNWGZSVANLYSJR
|
6.8 | IC50 | 2 | — | |
GGWWZSKHPHUDIG
|
6.8 | IC50 | 4 | — | |
JJFSLRIQURRAOH
|
6.8 | IC50 | 4 | — | |
NOMZQLLANMQZNR
|
6.8 | IC50 | 4 | — | |
NOMZQLLANMQZNR
|
6.8 | IC50 | 4 | — | |
YGOOSESWCCPOHN
|
6.8 | IC50 | 4 | — | |
LKKLTPUNQSFPCU
|
6.8 | IC50 | 3 | — | |
UOEMJLRQPFDRNW
|
6.8 | IC50 | 2 | — | |
DUDURFQIJNZVOS
|
6.8 | Ki | 2 | — | |
FJKPOCSUBVDARQ
|
6.8 | IC50 | 3 | — | |
OLIMBXKACVCIMM
|
6.8 | IC50 | 3 | — | |
ZRXIUMYAXSVUSM
|
6.8 | Ki | 2 | — | |
WTCANZGRFGLWSN
|
6.8 | IC50 | 3 | — | |
PBHZOHMBRYRIGB
|
6.8 | IC50 | 2 | — | |
GCWIICJLIHIUNY
|
6.7 | IC50 | 7 | — | |
JSXZJHBCLGHLND
|
6.7 | Ki | 3 | — | |
LWTLVKKUNGVFHE
|
6.7 | IC50 | 2 | — | |
OZAFFYABJNEFEY
|
6.7 | Ki | 2 | — |