Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WFIHUJGSDBPSIV
|
7.1 | Ki | 2 | — | |
GZGBHAIADJLADQ
|
7.1 | IC50 | 4 | — | |
QYTUQGRZRZIUCK
|
7.1 | Ki | 2 | — | |
FENBNSNVOOUUMD
|
7.1 | Ki | 3 | — | |
FENBNSNVOOUUMD
|
7.1 | Ki | 3 | — | |
FKWDMIPLXKTQTC
|
7.1 | IC50 | 2 | — | |
IRZHJAGVDPAPOG
|
7.1 | Ki | 3 | — | |
QZBJWYBUXVGFSV
|
7.1 | Ki | 3 | — | |
SRQKADSCZJGWOI
|
7.1 | IC50 | 2 | — | |
FXILBKWGQQHVJE
|
7.1 | IC50 | 2 | — | |
KIDPFKMKRUSRRX
|
7.1 | IC50 | 4 | — | |
HFYVNXIFHUNOBW
|
7.1 | IC50 | 2 | — | |
IVVYCBBKQYBPIG
|
7.1 | IC50 | 2 | — | |
QLCDJMHVAVRDAU
|
7.1 | Ki | 3 | — | |
BVKBZERLIAEOOG
|
7.1 | Ki | 2 | — | |
SIIJWJNEODXHNY
|
7.1 | IC50 | 7 | — | |
MFKDQBYQJMCGMB
|
7.0 | Ki | 2 | — | |
SVWMYRNQZSRCPR
|
7.0 | IC50 | 2 | — | |
WAWCVPQCGNEDNX
|
7.0 | IC50 | 4 | — | |
YLWGTLCVWLJFOC
|
7.0 | IC50 | 2 | — | |
XTQBGGSWYJPJBX
|
7.0 | Ki | 2 | — | |
KKKHMKQUVHHTJX
|
7.0 | Ki | 4 | — | |
VZTRAYHUTKYOCB
|
7.0 | IC50 | 4 | — | |
ZAJWZYOGSAVOOQ
|
7.0 | Ki | 2 | — | |
AWOBKJOFJAEFMO
|
7.0 | IC50 | 3 | — | |
DQSSVNLGIWUXRQ
|
7.0 | IC50 | 4 | — | |
DTKJGQRHUHIVHR
|
7.0 | IC50 | 3 | — | |
FNKYIUJUGBJYQM
|
7.0 | IC50 | 3 | — | |
GFBNAICZWORTRP
|
7.0 | IC50 | 3 | — | |
HFXHAUDVMVAJNA
|
7.0 | IC50 | 3 | — | |
HJUPPNTXGDFNAO
|
7.0 | IC50 | 3 | — | |
JOXOPPDPWDHDAQ
|
7.0 | IC50 | 2 | — | |
LTCAMZPTBRHGIT
|
7.0 | IC50 | 4 | — | |
LTEDERVMQUPCSO
|
7.0 | IC50 | 3 | — | |
MMOPUWHYSSYPDF
|
7.0 | IC50 | 2 | — | |
NEFVERIOUCVCKE
|
7.0 | IC50 | 3 | — | |
NGAUZCRIRRLFOO
|
7.0 | IC50 | 3 | — | |
OEGLOMHKABJFTM
|
7.0 | IC50 | 2 | — | |
PHDAPWSITYILFC
|
7.0 | IC50 | 2 | — | |
TXGCKASBHJKJOM
|
7.0 | Ki | 2 | — | |
UTNIKRVBYGTXDR
|
7.0 | IC50 | 2 | — | |
ZZDKLZGEJYCCFB
|
7.0 | IC50 | 4 | — | |
ZZDKLZGEJYCCFB
|
7.0 | IC50 | 4 | — | |
DQAYLGVDWYKLKW
|
7.0 | Ki | 2 | — | |
HGAFZDAZAKRDKS
|
7.0 | IC50 | 2 | — | |
LGACDLUVLNDBOB
|
7.0 | IC50 | 4 | — | |
USPHVRZFPMWSPR
|
7.0 | IC50 | 4 | — | |
FIFIFHHKQXWADB
|
7.0 | IC50 | 3 | — | |
HIIHCLZTHBBBAH
|
7.0 | Ki | 3 | — | |
JYBPZVHLFOMEHP
|
7.0 | Ki | 3 | — |