Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CCFPTWLGKMFRNV
|
7.3 | IC50 | 2 | — | |
OGWCUAHSOGTYTL
|
7.3 | Ki | 2 | — | |
VAIIZXKEFCDOFC
|
7.3 | IC50 | 2 | — | |
VLZYXSQGILGQAI
|
7.3 | IC50 | 6 | — | |
IGBRTMNMZLDZHD
|
7.3 | IC50 | 2 | — | |
QCZGUQGVICOTKX
|
7.3 | IC50 | 3 | — | |
QCZGUQGVICOTKX
|
7.3 | IC50 | 4 | — | |
BQWWAZOZDJROFE
|
7.3 | IC50 | 4 | — | |
HSECIQLWCNQZCS
|
7.3 | Ki | 2 | — | |
HZRCZFGJFFPTAI
|
7.3 | IC50 | 2 | — | |
OZNGVEHEJAXJKC
|
7.3 | Ki | 3 | — | |
RLOIWJYMAZZFLS
|
7.3 | Ki | 3 | — | |
JEBQNHANRCYVLC
|
7.3 | IC50 | 4 | — | |
VPDWNQHHCKCYRB
|
7.3 | Ki | 2 | — | |
KTIQHTPWWOJKML
|
7.3 | Ki | 2 | — | |
YRVGOKKZUPVDNC
|
7.3 | IC50 | 3 | — | |
ZEXMBYOEZWSCKY
|
7.3 | IC50 | 3 | — | |
BNUJXKLKLWZLCQ
|
7.2 | IC50 | 2 | — | |
RBTCEAUSBIXELN
|
7.2 | IC50 | 2 | — | |
TXNDJCXNKMIHRP
|
7.2 | Ki | 3 | — | |
YBSWDIITMXRJIB
|
7.2 | IC50 | 4 | — | |
ABTLMVRXRICKRX
|
7.2 | IC50 | 3 | — | |
JPASHDRVAQOCBT
|
7.2 | Ki | 2 | — | |
YMDHLHZVVIBPIA
|
7.2 | IC50 | 3 | — | |
ROKVPWHHBYTRKM
|
7.2 | IC50 | 2 | — | |
DOCKONDCDYZCFE
|
7.2 | IC50 | 3 | — | |
JOOITSNPEJONKV
|
7.2 | Ki | 2 | — | |
ROYHQNKYCLIWRK
|
7.2 | IC50 | 2 | — | |
WAGDARZNQCGUPI
|
7.2 | IC50 | 2 | — | |
BPIZQAAUSWBFNS
|
7.2 | IC50 | 4 | — | |
BPIZQAAUSWBFNS
|
7.2 | IC50 | 4 | — | |
MBRJRDMYBURHPH
|
7.2 | IC50 | 2 | — | |
RSEOJELKUSEFQD
|
7.2 | IC50 | 4 | — | |
HAPWVSXVFDZFLG
|
7.2 | Ki | 2 | — | |
INIJDZXPDCZFFR
|
7.2 | IC50 | 2 | — | |
NTPPZLBAUWCCNL
|
7.2 | IC50 | 2 | — | |
BNXDYZBRHZMVRA
|
7.2 | IC50 | 4 | — | |
ANZFZARZEQENJQ
|
7.2 | Ki | 4 | — | |
MTLWLBWTUSPBQE
|
7.2 | IC50 | 2 | — | |
OQVJUAAFCYLUII
|
7.2 | IC50 | 4 | — | |
SWDBTDNRUQLZFB
|
7.2 | Ki | 2 | — | |
TYRKGQFUSLPRSY
|
7.2 | IC50 | 4 | — | |
VOROYGUSPRVWST
|
7.2 | Ki | 3 | — | |
BHVRFNJEHAGAIV
|
7.2 | IC50 | 4 | — | |
HZJOEDHTKKTHRB
|
7.2 | IC50 | 3 | — | |
MQPFSCOBQLFTCQ
|
7.2 | IC50 | 2 | — | |
OQVCDUQURLATAT
|
7.2 | IC50 | 2 | — | |
LIQDTPYQUQZTGR
|
7.1 | Ki | 2 | — | |
LKVLCOTZWXWKQV
|
7.1 | IC50 | 2 | — | |
ZNUMRCPRXWDFHV
|
7.1 | IC50 | 4 | — |