Target Details
| UniProt AC | P43235 |
|---|---|
| Gene Symbol | CTSK |
| Protein Name | Cathepsin K |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 835
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (5)
Associated Diseases (2)
Active Molecules (835)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CAQLLDUOKIHSBN
|
11.5 | IC50 | 3 | — | |
HWNYTOPEHDSGOF
|
11.5 | IC50 | 3 | — | |
YWXWRCMYHIYBSJ
|
11.1 | Ki | 4 | — | |
YZBDFADJOLGKFN
|
11.1 | IC50 | 3 | — | |
LMZYZVWKTJFLSL
|
11.0 | Ki | 3 | — | |
UEZMKFGTDYYCKL
|
11.0 | IC50 | 3 | — | |
GASCFELIQZXIAB
|
11.0 | IC50 | 3 | — | |
JESRGSWARNNMLP
|
11.0 | Ki | 4 | — | |
LCGRTAPRJZMTIT
|
11.0 | IC50 | 3 | — | |
AKAUMTCIIOMDTI
|
10.9 | IC50 | 3 | — | |
CLOALCKDNZPWBO
|
10.8 | Ki | 4 | — | |
YCYQOGPWUSMXGX
|
10.7 | Ki | 4 | — | |
KFTMZNIURYIOKI
|
10.7 | Ki | 4 | — | |
VLROHFCAQABUTJ
|
10.7 | IC50 | 3 | — | |
UPWNNHRBMJWIBW
|
10.5 | IC50 | 3 | — | |
AUPZRAAKTGPDLC
|
10.5 | Ki | 4 | — | |
VCANIUOBHBAPJH
|
10.5 | Ki | 3 | — | |
BWYBBMQLUKXECQ
|
10.4 | Ki | 5 | — | |
ARWSHTCIMVGBCQ
|
10.3 | Ki | 4 | — | |
BEMWXCUECCHZDO
|
10.3 | IC50 | 4 | — | |
GZBOGFDHJAMENH
|
10.2 | Ki | 4 | — | |
SCCNQBNFEHNRCO
|
10.2 | Ki | 4 | — | |
MWBPTVRPPPPZPG
|
10.1 | Ki | 4 | — | |
NFPHFQIUODNJRD
|
10.1 | IC50 | 5 | — | |
HCERRVOHXYKRJP
|
10.0 | IC50 | 2 | — | |
QBAMPEZJGKYTHV
|
10.0 | IC50 | 3 | — | |
LRGPAVMYPWWORG
|
10.0 | Ki | 4 | — | |
PGGUOGKHUUUWAF
|
10.0 | IC50 | 3 | — | |
ULFKHVBAISSIOJ
|
10.0 | IC50 | 4 | — | |
QQPGHYGBHVMSNJ
|
9.9 | IC50 | 3 | — | |
FTJHEEIVOBBMMC
|
9.8 | Ki | 5 | — | |
MCKCVIDASJTQSU
|
9.8 | Ki | 3 | — | |
XWMOCHXKDCBQPV
|
9.8 | Ki | 4 | — | |
ONHOINLCWRTXCR
|
9.7 | Ki | 2 | — | |
FWIVDMJALNEADT
|
9.7 | IC50 | 5 | — | |
GNPSTHRVAFKOMP
|
9.7 | IC50 | 2 | — | |
LWTHIEWNFZTHDQ
|
9.7 | IC50 | 4 | — | |
OANFHMRTEKMMQQ
|
9.7 | IC50 | 2 | — | |
SVLOPEXSNUUHTH
|
9.7 | IC50 | 3 | — | |
VEZZBPBPTOZPBS
|
9.7 | IC50 | 5 | — | |
VYFDSJLOCIGIKP
|
9.7 | IC50 | 3 | — | |
YEQBMHWVACZUNK
|
9.7 | IC50 | 3 | — | |
ATHIBBJHLIDXBN
|
9.5 | IC50 | 2 | — | |
BHXUXLQVSXLWEI
|
9.5 | IC50 | 3 | — | |
FQZHBMQEEUCQNE
|
9.5 | IC50 | 3 | — | |
HSRNAGMZGLYZKO
|
9.5 | IC50 | 3 | — | |
MJJJUBXJMQFNNM
|
9.5 | IC50 | 3 | — | |
MQVPDECTVKAJFG
|
9.5 | IC50 | 3 | — | |
STBKPRWJLMIORW
|
9.5 | IC50 | 3 | — | |
ZQXYZTRTLGOBEJ
|
9.5 | IC50 | 4 | — |