Target Details
| UniProt AC | P43220 |
|---|---|
| Gene Symbol | GLP1R |
| Protein Name | Glucagon-like peptide 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 6.84
KEGG Pathways (4)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CBVCZFGXHXORBI
|
9.9 | IC50 | 6 | — | |
OQWWPGFZOFJMCP
|
7.6 | IC50 | 3 | — | |
QVSVLRYVPXFJOT
|
7.0 | IC50 | 3 | — | |
MREMAWQXBDPMKX
|
7.0 | IC50 | 3 | — | |
UEOWVVNOBYAFMV
|
6.8 | IC50 | 2 | — | |
FMOBKUHELCHCKY
|
6.5 | IC50 | 2 | — | |
MFEIZMHODFOWAT
|
6.2 | IC50 | 2 | — | |
XIKBNACNRMHVLD
|
6.2 | IC50 | 2 | — | |
PFOUJNFXNRYXCU
|
6.1 | IC50 | 2 | — | |
ZBMZGBGZOQFXEP
|
6.1 | Ki | 3 | — | |
BZXMLCVDKDXRQY
|
6.0 | IC50 | 11 | — |