Target Details
| UniProt AC | P43119 |
|---|---|
| Gene Symbol | PTGIR |
| Protein Name | Prostacyclin receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 22
- Clinical molecules 0
- Avg pChEMBL 6.95
KEGG Pathways (3)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XQSDEHHCLDLVST
|
8.2 | Ki | 2 | — | |
XQSDEHHCLDLVST
|
8.2 | Ki | 2 | — | |
HIFJCPQKFCZDDL
|
8.1 | IC50 | 5 | — | |
NPDKXVKJRHPDQT
|
8.0 | IC50 | 4 | — | |
UMQLASXGJFGXFL
|
8.0 | IC50 | 3 | — | |
ARUGKOZUKWAXDS
|
7.8 | Ki | 3 | — | |
XECAIYOLUPUKEJ
|
7.4 | Ki | 3 | — | |
XRISENIKJUKIHD
|
7.4 | IC50 | 2 | — | |
XZFRIPGNUQRGPI
|
7.2 | Ki | 7 | — | |
PAYNQYXOKJDXAV
|
6.8 | IC50 | 2 | — | |
CSDQJTVCSKACSP
|
6.8 | Ki | 2 | — | |
RFHFLABUEIMYLC
|
6.7 | Ki | 2 | — | |
XEYBRNLFEZDVAW
|
6.6 | IC50 | 7 | — | |
XSQAICBCYIFUQS
|
6.4 | Ki | 5 | — | |
PNUIFGGEAVOVPQ
|
6.4 | Ki | 2 | — | |
VQNGUZVGSDDDEI
|
6.3 | Ki | 2 | — | |
SDGUUEATIIAOTG
|
6.2 | Ki | 2 | — | |
VIPZGFVAWMFKDS
|
6.2 | Ki | 2 | — | |
DCYHRPUPJCRAGG
|
6.2 | Ki | 9 | — | |
PXFUYKMANFDTAA
|
6.1 | Ki | 2 | — | |
UQAGCAUWYZNISV
|
6.1 | Ki | 2 | — | |
PUQLADUSPHHAJY
|
6.0 | IC50 | 2 | — |