Target Details
| UniProt AC | P43088 |
|---|---|
| Gene Symbol | PTGFR |
| Protein Name | Prostaglandin F2-alpha receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 23
- Clinical molecules 0
- Avg pChEMBL 7.47
KEGG Pathways (3)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VJGGHXVGBSZVMZ
|
8.8 | IC50 | 3 | — | |
FAPQZCFUFGJPFI
|
8.7 | IC50 | 4 | — | |
VJGGHXVGBSZVMZ
|
8.7 | IC50 | 3 | — | |
WWSWYXNVCBLWNZ
|
8.6 | Ki | 2 | — | |
CHDOVUGJRCWTAC
|
8.5 | IC50 | 2 | — | |
TUXFWOHFPFBNEJ
|
8.2 | Ki | 3 | — | |
PXGPLTODNUVGFL
|
8.2 | IC50 | 4 | — | |
KVSLCHMLOXAYQJ
|
8.0 | IC50 | 2 | — | |
CCIGYTQGGWYUNA
|
7.9 | IC50 | 2 | — | |
PXGPLTODNUVGFL
|
7.9 | Ki | 7 | — | |
JGZRPRSJSQLFBO
|
7.7 | Ki | 2 | — | |
YTZPMGSDIYCPCW
|
7.5 | IC50 | 2 | — | |
RTPIJAVXJNAJOS
|
7.5 | IC50 | 2 | — | |
PTOJVMZPWPAXER
|
7.1 | Ki | 3 | — | |
XEYBRNLFEZDVAW
|
6.9 | Ki | 7 | — | |
UQZVCDCIMBLVNR
|
6.7 | Ki | 3 | — | |
LQANGKSBLPMBTJ
|
6.6 | Ki | 3 | — | |
XUWIMBOVFJGMEM
|
6.6 | IC50 | 2 | — | |
FJMQKJOWJVMHPQ
|
6.5 | Ki | 5 | — | |
XZFRIPGNUQRGPI
|
6.4 | Ki | 7 | — | |
NZGFSDWJUZOAAX
|
6.3 | Ki | 6 | — | |
SOONLSMFDWIFKR
|
6.2 | IC50 | 2 | — | |
HIFJCPQKFCZDDL
|
6.2 | Ki | 5 | — |