Target Details
| UniProt AC | P43003 |
|---|---|
| Gene Symbol | SLC1A3 |
| Protein Name | Excitatory amino acid transporter 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00375 (SDF) |
Summary
- Multi-target molecules 28
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (28)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKWBPFZLNZBTPN
|
8.3 | IC50 | 3 | — | |
JBOQCANANDNLOB
|
8.2 | IC50 | 3 | — | |
LPWONNPEPDHEAI
|
8.1 | IC50 | 3 | — | |
VQNZVGSJHAMMFA
|
8.0 | IC50 | 3 | — | |
RPXRQPZQCZLBCH
|
7.9 | IC50 | 3 | — | |
YYNRJPQKRZAORR
|
7.7 | IC50 | 3 | — | |
RSBUOFNPLDYKRF
|
7.5 | IC50 | 3 | — | |
NGYBWUWAZHMQRP
|
7.0 | IC50 | 3 | — | |
VNESGVWLCUTKMJ
|
7.0 | IC50 | 3 | — | |
XADHWMPKONEAES
|
6.9 | IC50 | 2 | — | |
OXLGRRCHUJEPLH
|
6.9 | IC50 | 3 | — | |
WXVBLLQGBPMCBA
|
6.8 | IC50 | 3 | — | |
FAAZYFWXJOLYDB
|
6.7 | IC50 | 3 | — | |
UJOVSQYLMTYASM
|
6.7 | IC50 | 3 | — | |
HJLWSVGVNAASDU
|
6.5 | IC50 | 3 | — | |
QDIIRLCSVINDSC
|
6.5 | IC50 | 3 | — | |
UWHHZYOBBZGRIH
|
6.5 | IC50 | 3 | — | |
PHSLITQWZPTNLO
|
6.5 | IC50 | 2 | — | |
AGGLVRRXRHFAJT
|
6.5 | IC50 | 3 | — | |
CPAPJLPIAMJYMZ
|
6.4 | IC50 | 2 | — | |
MJVRZPPTZDJHOD
|
6.4 | IC50 | 3 | — | |
FKSWJLRIKQYTFH
|
6.2 | IC50 | 2 | — | |
MBQGVKLYPFNSIW
|
6.2 | IC50 | 3 | — | |
WZYMCYMJMKQWQX
|
6.2 | IC50 | 2 | — | |
JSERPLUABIILRN
|
6.1 | IC50 | 2 | — | |
BNYDDAAZMBUFRG
|
6.1 | IC50 | 2 | — | |
ZUJCVROZZWXJLM
|
6.0 | IC50 | 3 | — | |
ZWSCZNCTZIFFBX
|
6.0 | IC50 | 2 | — |