Target Details
| UniProt AC | P42685 |
|---|---|
| Gene Symbol | FRK |
| Protein Name | Tyrosine-protein kinase FRK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 234
- Clinical molecules 36
- Avg pChEMBL 7.03
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YABJJWZLRMPFSI
|
6.2 | Kd | 34 | — | |
YMSXHRWUGLAAKL
|
6.2 | IC50 | 14 | Yes | |
HEUSUIRCBWROMH
|
6.2 | Ki | 64 | — | |
UPYHVTCMTMZKAX
|
6.2 | Ki | 12 | — | |
WDTHDWKPTWWHLS
|
6.2 | IC50 | 13 | — | |
BFSMGDJOXZAERB
|
6.1 | Kd | 33 | — | |
LCVIRAZGMYMNNT
|
6.1 | Kd | 20 | — | |
XXJWYDDUDKYVKI
|
6.1 | Kd | 52 | — | |
FLBNLJLONKAPLR
|
6.1 | Kd | 31 | — | |
UIARLYUEJFELEN
|
6.1 | Kd | 289 | Yes | |
ZCCPLJOKGAACRT
|
6.1 | Kd | 599 | — | |
CUIHSIWYWATEQL
|
6.1 | Kd | 61 | Yes | |
CLRFYTGANQZOBS
|
6.1 | Ki | 41 | — | |
CSGQVNMSRKWUSH
|
6.1 | Kd | 21 | — | |
IOBVCHJTLVPPBR
|
6.1 | Ki | 39 | — | |
JCZBWICLNFNCMR
|
6.1 | Ki | 9 | — | |
NXNQLECPAXXYTR
|
6.1 | Ki | 29 | — | |
PEEMSUJXJVLHFP
|
6.1 | Ki | 4 | — | |
YUOWJICKAJQZLS
|
6.1 | Ki | 35 | — | |
ZQUSFAUAYSEREK
|
6.1 | Ki | 7 | — | |
DKNUPRMJNUQNHR
|
6.1 | Kd | 33 | — | |
AQQWWOMMPDCTLW
|
6.0 | Ki | 10 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTEIFNKAUNYNJU
|
6.0 | IC50 | 114 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NRSGWEVTVGZDFC
|
6.0 | Ki | 50 | — | |
OPLHMHMCXQXEQG
|
6.0 | Ki | 10 | — | |
OUJZYQBEFNDJQN
|
6.0 | Ki | 71 | — | |
PKCDDUHJAFVJJB
|
6.0 | Ki | 13 | — | |
QAJPIJHWTGPUNZ
|
6.0 | Ki | 37 | — | |
QONPPIZSNSSCSK
|
6.0 | Ki | 45 | Yes | |
RIUZPIBUSOHUKF
|
6.0 | Ki | 23 | — | |
YDOPLCNFRXOHCC
|
6.0 | Ki | 28 | — |