Target Details
| UniProt AC | P42685 |
|---|---|
| Gene Symbol | FRK |
| Protein Name | Tyrosine-protein kinase FRK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 234
- Clinical molecules 36
- Avg pChEMBL 7.03
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AAKJLRGGTJKAMG
|
6.5 | Ki | 50 | Yes | |
BHSOPYVVEZFHDB
|
6.5 | Ki | 25 | Yes | |
BSFNGHCTZDCQBF
|
6.5 | Ki | 93 | — | |
HHHWHXLLZCRLAO
|
6.5 | Ki | 5 | — | |
KTUFNOKKBVMGRW
|
6.5 | Ki | 38 | Yes | |
MFMXAWQGPQXDRJ
|
6.5 | Ki | 27 | — | |
NLUPJKQOKWBWFC
|
6.5 | Ki | 69 | — | |
YCOYDOIWSSHVCK
|
6.5 | Ki | 10 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
VNBRGSXVFBYQNN
|
6.5 | Kd | 22 | Yes | |
AHBFBRPGNOVEBK
|
6.4 | IC50 | 11 | — | |
MVCOAUNKQVWQHZ
|
6.4 | Kd | 54 | Yes | |
WVUNYSQLFKLYNI
|
6.4 | Kd | 46 | Yes | |
OSVUGUHRKMMBSE
|
6.4 | Kd | 170 | — | |
RNOAOAWBMHREKO
|
6.4 | IC50 | 15 | — | |
DILZQOYOWSNWDQ
|
6.4 | Ki | 2 | — | |
DJLORVJVWIBDME
|
6.4 | Ki | 24 | — | |
FUMCKNCUEAQHCV
|
6.4 | Ki | 103 | — | |
GUMBHNMWKMFKRT
|
6.4 | Ki | 23 | — | |
HEKAIDKUDLCBRU
|
6.4 | Ki | 20 | — | |
ISVHLTLEHRZKJC
|
6.4 | Ki | 19 | — | |
LVECPYVAIBNSRV
|
6.4 | Ki | 33 | — | |
MPVGZUGXCQEXTM
|
6.4 | Kd | 61 | Yes | |
MTCHQDWUHQADSY
|
6.4 | Ki | 29 | — | |
PYDWRLNPMMKKCI
|
6.4 | Ki | 7 | — | |
RTDSHUGNRVXRHN
|
6.4 | Ki | 51 | — | |
TUJUZVJICDSNLY
|
6.4 | Ki | 19 | — | |
XBAIEEJJCJHBDL
|
6.4 | Ki | 17 | — | |
XYZNKCSDQRKAFR
|
6.4 | Ki | 53 | — | |
ZKHDDJKHTPLPOQ
|
6.4 | Ki | 62 | — | |
ZPXPEKQMLOAPLT
|
6.4 | Ki | 15 | — | |
ZGBAJMQHJDFTQJ
|
6.4 | Kd | 15 | — | |
VTJHGMZHVOXJPG
|
6.3 | IC50 | 15 | — | |
ADMFLILDQJSEIK
|
6.3 | Ki | 72 | — | |
FGWOKLCRQJXPPQ
|
6.3 | Ki | 14 | — | |
IGGNAIYXGIUMQZ
|
6.3 | Ki | 5 | — | |
NERQMDXDVAZVNX
|
6.3 | Ki | 13 | — | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
MLDQJTXFUGDVEO
|
6.3 | Kd | 85 | Yes | |
OSAWFUCUZJNEID
|
6.3 | IC50 | 20 | — | |
WINHZLLDWRZWRT
|
6.3 | Kd | 201 | Yes | |
WMMNTQFZCHUZSM
|
6.3 | IC50 | 14 | — | |
DPZGKYJHTOSMIA
|
6.3 | IC50 | 8 | — | |
IBCGPVVKHZXWNX
|
6.3 | IC50 | 7 | — | |
KUCNBQPAJZRQMJ
|
6.3 | IC50 | 11 | — | |
MJQGHLODJHABRA
|
6.3 | IC50 | 10 | — | |
QZCWPDPWSBOTEU
|
6.3 | IC50 | 7 | — | |
VWDNDBICKRVFCP
|
6.3 | IC50 | 4 | — | |
ONIQOQHATWINJY
|
6.2 | Kd | 25 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes |