Target Details
| UniProt AC | P42685 |
|---|---|
| Gene Symbol | FRK |
| Protein Name | Tyrosine-protein kinase FRK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 234
- Clinical molecules 36
- Avg pChEMBL 7.03
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXHOCWWJSGCZLC
|
7.1 | Ki | 18 | — | |
UOVCGJXDGOGOCZ
|
7.1 | Ki | 59 | — | |
XFWUTMHVDGPWLH
|
7.1 | Ki | 75 | — | |
XYFPWWZEPKGCCK
|
7.1 | IC50 | 34 | — | |
ZGZVRPRSFXRGCF
|
7.1 | Ki | 76 | — | |
ZVWRFVCNQOECJS
|
7.1 | Ki | 71 | — | |
HHZIURLSWUIHRB
|
7.1 | Kd | 57 | Yes | |
LSJWYMSFUWBGPN
|
7.1 | IC50 | 17 | — | |
WJEOLQLKVOPQFV
|
7.1 | Kd | 24 | — | |
CNTCGRJDUJEUDG
|
7.0 | Ki | 37 | — | |
RAHBGWKEPAQNFF
|
7.0 | Kd | 26 | — | |
YEKVTSRZMPLPFK
|
7.0 | Ki | 17 | — | |
ZLHFILGSQDJULK
|
7.0 | Ki | 37 | Yes | |
JUSWPUDQOKINJO
|
7.0 | IC50 | 16 | — | |
XKFTZKGMDDZMJI
|
7.0 | Kd | 64 | Yes | |
GZGRGXPFYDFNHF
|
6.9 | Kd | 3 | — | |
DBXGGXLBTWZXBB
|
6.9 | Ki | 39 | — | |
DLWMVUDMPMKGEE
|
6.9 | Ki | 24 | — | |
GWMATETWMAQOFL
|
6.9 | Ki | 36 | — | |
HXHAJRMTJXHJJZ
|
6.9 | Kd | 52 | Yes | |
MGGBYMDAPCCKCT
|
6.9 | IC50 | 23 | — | |
RQJIDUOCLNMUHR
|
6.9 | Ki | 15 | — | |
UDFDIIVNIYWXDM
|
6.9 | Ki | 74 | — | |
WINHZLLDWRZWRT
|
6.9 | Ki | 66 | — | |
GZYUJXFTHLKPAK
|
6.9 | IC50 | 16 | — | |
SPMVMDHWKHCIDT
|
6.8 | Kd | 30 | — | |
OPHSZSZDICRBPP
|
6.8 | IC50 | 16 | — | |
OMIQRSKHABIPRH
|
6.8 | IC50 | 15 | — | |
BOBGABAXWFYHQX
|
6.8 | Ki | 9 | — | |
FAYAUAZLLLJJGH
|
6.8 | Ki | 36 | Yes | |
GDYZFFBMSBDTAA
|
6.8 | Ki | 60 | — | |
PCQMERRARZKTPW
|
6.8 | Ki | 68 | — | |
QXRJBJVCBQSLTA
|
6.8 | Ki | 29 | — | |
RYAVJHIPOWNWDE
|
6.8 | Ki | 38 | — | |
UHTHHESEBZOYNR
|
6.8 | Kd | 66 | Yes | |
VWMJHAFYPMOMGF
|
6.8 | Kd | 15 | — | |
XYFZVVYVIFJBIS
|
6.7 | IC50 | 17 | — | |
JOOXLOJCABQBSG
|
6.7 | Kd | 139 | — | |
XLFYOIVELARSKP
|
6.7 | Ki | 33 | — | |
LAUHLGUSVSJYCI
|
6.7 | IC50 | 16 | — | |
WKDACQVEJIVHMZ
|
6.7 | Kd | 46 | — | |
ACNCCUVYXQGPKZ
|
6.6 | Ki | 31 | — | |
CDMGBJANTYXAIV
|
6.6 | Ki | 34 | Yes | |
CQFVDHNTTRWVQD
|
6.6 | Ki | 9 | — | |
GMYYMEOGFRKSFS
|
6.6 | Ki | 29 | — | |
KTEIFNKAUNYNJU
|
6.6 | Ki | 48 | — | |
MADCXGNPDBWPLM
|
6.6 | Ki | 25 | — | |
TVLFEDKEAOXRCZ
|
6.6 | Ki | 22 | — | |
XGALLCVXEZPNRQ
|
6.6 | Ki | 39 | Yes | |
SHPFDGWALWEPGS
|
6.5 | Kd | 35 | — |