Target Details
| UniProt AC | P42685 |
|---|---|
| Gene Symbol | FRK |
| Protein Name | Tyrosine-protein kinase FRK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 234
- Clinical molecules 36
- Avg pChEMBL 7.03
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ODPGGGTTYSGTGO
|
7.6 | Kd | 153 | — | |
QQWUGDVOUVUTOY
|
7.6 | Kd | 231 | Yes | |
DSZLKOXKYRREEO
|
7.5 | IC50 | 10 | — | |
DYSRECIVMDGUQU
|
7.5 | Ki | 29 | — | |
GCYXEGSPUDSZJY
|
7.5 | Ki | 82 | — | |
GXJSLIOOPZRPEV
|
7.5 | Ki | 34 | — | |
JXNMCDLXYWQTIW
|
7.5 | Ki | 13 | — | |
NFMGZVPRGVERNN
|
7.5 | Ki | 44 | — | |
SEVCBWKJSOLMNQ
|
7.5 | Ki | 38 | — | |
SPMHGQZFMNZCBV
|
7.5 | Ki | 30 | Yes | |
VLEFVPMCVJDTHZ
|
7.5 | Ki | 13 | — | |
XKZQZMSAWVDRSP
|
7.5 | Ki | 39 | Yes | |
YMIJUBCSOKSFRU
|
7.5 | Ki | 87 | — | |
SRSQULBCTWSVKL
|
7.5 | IC50 | 15 | — | |
FUZSHLVNKZZEKR
|
7.4 | IC50 | 16 | — | |
WVXNSAVVKYZVOE
|
7.4 | IC50 | 92 | — | |
BLQYVHBZHAISJM
|
7.4 | Ki | 54 | — | |
DJRPFIWIDKXORZ
|
7.4 | Ki | 9 | — | |
DZSUJUOJJJCWGG
|
7.4 | Ki | 55 | Yes | |
MZDKLVOWGIOKTN
|
7.4 | Ki | 80 | — | |
NRGYZNJPCGRCLV
|
7.4 | Ki | 52 | — | |
OWFXKTOLFUQPDJ
|
7.4 | Ki | 36 | — | |
UWDBNTXEKYRMSG
|
7.4 | Ki | 26 | — | |
XNEPVLVYFUGJLF
|
7.4 | Ki | 27 | — | |
YEHCNYAQEBQCCS
|
7.4 | Ki | 74 | — | |
PTHVKCSYXICMAR
|
7.4 | IC50 | 14 | — | |
HKSZLNNOFSGOKW
|
7.3 | Kd | 408 | — | |
HKSZLNNOFSGOKW
|
7.3 | Kd | 213 | — | |
CDISOBGWDHAHGF
|
7.3 | IC50 | 16 | — | |
DKSNLQYRZJKYOC
|
7.3 | Ki | 51 | — | |
LCGSWTFWYNYUKS
|
7.3 | Ki | 26 | — | |
LGHBDVLAHHANMX
|
7.3 | Ki | 53 | — | |
MHCPAORAYMTGCZ
|
7.3 | Ki | 37 | — | |
RWEHAHIEUDLKGT
|
7.3 | Ki | 33 | — | |
WPXVVAWAHQHJPF
|
7.3 | IC50 | 41 | — | |
AILRADAXUVEEIR
|
7.3 | IC50 | 75 | — | |
IIXWYSCJSQVBQM
|
7.3 | IC50 | 18 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 15 | — | |
VXYZCOCRVAQWBG
|
7.3 | IC50 | 15 | — | |
NJKRMPNUGZAMJN
|
7.3 | IC50 | 5 | — | |
PGQWALGGBUYLQF
|
7.2 | IC50 | 12 | — | |
ADLPKFFMGIJZIM
|
7.2 | Ki | 44 | — | |
BIKYDWLMTPRSQL
|
7.2 | Ki | 50 | — | |
GCBJDOWIQHMCMR
|
7.2 | Ki | 84 | — | |
KRIUNPBAQZGFQA
|
7.2 | Ki | 76 | — | |
LYNBNVBMAGDJRW
|
7.2 | Ki | 81 | — | |
YEPNVBNYCRGZRX
|
7.2 | Ki | 26 | — | |
NHHQJBCNYHBUSI
|
7.2 | Kd | 220 | — | |
GEGCXGMFUYJULA
|
7.1 | Ki | 30 | Yes | |
RYYNGWLOYLRZLK
|
7.1 | Ki | 104 | — |