Target Details
| UniProt AC | P42685 |
|---|---|
| Gene Symbol | FRK |
| Protein Name | Tyrosine-protein kinase FRK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 234
- Clinical molecules 36
- Avg pChEMBL 7.03
Active Molecules (234)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
9.5 | Kd | 102 | Yes | |
AQSSMEORRLJZLU
|
9.0 | Kd | 34 | Yes | |
CFIBXVQLBVNOHW
|
9.0 | Ki | 64 | — | |
OWRXHGAFWZFFCW
|
9.0 | Ki | 113 | — | |
XKFTZKGMDDZMJI
|
8.9 | Ki | 56 | — | |
PHXJVRSECIGDHY
|
8.9 | IC50 | 59 | — | |
WFTZMAAMCVPJJT
|
8.7 | Ki | 26 | — | |
WPHKIQPVPYJNAX
|
8.7 | Ki | 81 | — | |
UBPYILGKFZZVDX
|
8.7 | Kd | 130 | Yes | |
XCHWBXBDZRJVDP
|
8.6 | Ki | 51 | — | |
XOOAAYRIVATZNM
|
8.6 | Ki | 55 | — | |
CXBBWVXSZINRCS
|
8.5 | Ki | 41 | — | |
RBXYGQNZRVPDNB
|
8.5 | Ki | 34 | — | |
UUWNXFJBBYAMDT
|
8.5 | Ki | 46 | — | |
ZVPDNRVYHLRXLX
|
8.5 | Ki | 35 | Yes | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
VMOVZKURWYNTLN
|
8.4 | Ki | 7 | — | |
VAARYSWULJUGST
|
8.4 | Kd | 119 | Yes | |
PTVPBWWDGZSEAF
|
8.3 | Ki | 63 | — | |
VKBFHTIUXUCYRQ
|
8.3 | Ki | 66 | — | |
XJSFDMGICAWQFS
|
8.3 | Ki | 60 | — | |
XKZINYYXWJEYEL
|
8.3 | Ki | 37 | — | |
CIGMIXWAESLRNR
|
8.2 | Kd | 5 | — | |
UOOZSMNSBYVUGZ
|
8.2 | Ki | 32 | — | |
ZXLFIHLBHMLHFJ
|
8.1 | Ki | 31 | — | |
AIQDZMUPVYDVLB
|
8.0 | Ki | 48 | — | |
JZTOUVBEZONDKA
|
8.0 | Ki | 80 | — | |
CXQHYVUVSFXTMY
|
8.0 | Kd | 154 | — | |
OIANGKGOYKDGQV
|
7.9 | Kd | 10 | — | |
ZWVZORIKUNOTCS
|
7.9 | Ki | 69 | — | |
HAYYBYPASCDWEQ
|
7.8 | Ki | 47 | — | |
JSDGKSMNPHJDFK
|
7.8 | Ki | 35 | — | |
MOSKATHMXWSZTQ
|
7.8 | IC50 | 16 | Yes | |
MULNSLQVKKUPJN
|
7.8 | Ki | 41 | — | |
MVJMMLFMPWITEJ
|
7.8 | Ki | 110 | — | |
ULMCFLZUGRSEQA
|
7.8 | Ki | 17 | — | |
ZGDSBEUMPIMXBM
|
7.8 | Ki | 42 | — | |
YHVHYWYQEFELOW
|
7.7 | IC50 | 44 | — | |
HCNIBOQWDVOZKF
|
7.7 | Ki | 26 | — | |
PUPCRRRSBUYJAD
|
7.7 | Ki | 44 | Yes | |
QKPLUKMJEKRAJD
|
7.7 | Ki | 30 | Yes | |
UYJNQQDJUOUFQJ
|
7.7 | Ki | 68 | — | |
NZJCXRPMZJGVCC
|
7.7 | Kd | 8 | — | |
GQGMUKOYILWOIQ
|
7.6 | Ki | 25 | — | |
NWAUBAGBGOPJLF
|
7.6 | Ki | 51 | Yes | |
QNUKRWAIZMBVCU
|
7.6 | Ki | 46 | — | |
SRUYMJRFVGLQDV
|
7.6 | Ki | 37 | — | |
XBYVOPRDASFDMY
|
7.6 | Ki | 42 | — | |
XHORJSJFHVABEA
|
7.6 | Ki | 49 | — | |
XYXLUJQBBIBJFV
|
7.6 | Ki | 36 | — |