Target Details
| UniProt AC | P42684 |
|---|---|
| Gene Symbol | ABL2 |
| Protein Name | Tyrosine-protein kinase ABL2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 202
- Clinical molecules 75
- Avg pChEMBL 6.99
KEGG Pathways (4)
Active Molecules (202)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RPRCCKYNDFQWHV
|
6.5 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
6.5 | Kd | 599 | — | |
FWVUUGWQEZWWHV
|
6.4 | IC50 | 6 | Yes | |
WVUNYSQLFKLYNI
|
6.4 | Kd | 46 | Yes | |
QQWUGDVOUVUTOY
|
6.4 | Kd | 231 | Yes | |
PTOVCSIEMQUGPX
|
6.4 | IC50 | 5 | Yes | |
KOFGCEDKGQUYDQ
|
6.4 | IC50 | 6 | Yes | |
TWUSYQHQSFRUMW
|
6.4 | IC50 | 5 | Yes | |
WKDACQVEJIVHMZ
|
6.4 | Kd | 46 | — | |
SRWSCJJFUPPXPK
|
6.4 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.3 | Kd | 114 | — | |
PFTXFNSHFZLJNT
|
6.3 | IC50 | 17 | — | |
HNYSHAGTWNOVGB
|
6.3 | IC50 | 5 | Yes | |
NMGPNPSPONCMOZ
|
6.3 | IC50 | 3 | — | |
TUXRFGDOGJUGFD
|
6.3 | IC50 | 5 | Yes | |
UHEXEECCTNTZTE
|
6.3 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
6.3 | Kd | 200 | — | |
AGHOQYDPQAQJNL
|
6.3 | IC50 | 2 | — | |
ZWOJEBVNAWIFMO
|
6.3 | IC50 | 5 | Yes | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
IUHCHNLQYCBXNR
|
6.2 | IC50 | 5 | Yes | |
KKYWVNPRFIJNKB
|
6.2 | IC50 | 6 | Yes | |
HVXKQKFEHMGHSL
|
6.2 | Kd | 21 | — | |
NJLUOCLXYPXAHG
|
6.2 | IC50 | 3 | — | |
SEXVGHCKBMFFSZ
|
6.2 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
6.2 | Kd | 1075 | — | |
ZOROFBCOYYIWNJ
|
6.2 | IC50 | 5 | Yes | |
PHWPEULWFLWFAR
|
6.2 | IC50 | 3 | — | |
SRVDBASMNUCPHD
|
6.2 | IC50 | 5 | Yes | |
MJUOSFZKBYWVCP
|
6.2 | IC50 | 3 | — | |
RJBTYCBOXYRMMJ
|
6.2 | IC50 | 3 | — | |
UGGTXZIJVQPZJC
|
6.2 | IC50 | 3 | — | |
YXWFENMECIODNR
|
6.2 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
6.1 | Kd | 220 | — | |
UQRCJCNVNUFYDX
|
6.1 | Kd | 27 | — | |
XXJWYDDUDKYVKI
|
6.1 | Kd | 52 | — | |
KXHOCICVTKWLSA
|
6.1 | IC50 | 3 | — | |
OMZCMEYTWSXEPZ
|
6.1 | Kd | 43 | Yes | |
XISIJMIPHPQCQQ
|
6.1 | IC50 | 9 | — | |
IAYGCINLNONXHY
|
6.0 | Kd | 50 | — | |
ONIQOQHATWINJY
|
6.0 | Kd | 25 | — | |
XYFPWWZEPKGCCK
|
6.0 | Kd | 34 | — | |
AYCPARAPKDAOEN
|
6.0 | Kd | 73 | — | |
OSVUGUHRKMMBSE
|
6.0 | Kd | 170 | — | |
SHPFDGWALWEPGS
|
6.0 | Kd | 35 | — | |
IQMVMHITWPJRIL
|
6.0 | IC50 | 4 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
WGNQPAWFLWLKBL
|
6.0 | IC50 | 4 | Yes |