Target Details
| UniProt AC | P42684 |
|---|---|
| Gene Symbol | ABL2 |
| Protein Name | Tyrosine-protein kinase ABL2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 202
- Clinical molecules 75
- Avg pChEMBL 6.99
KEGG Pathways (4)
Active Molecules (202)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HYPPWDWGZRSMTQ
|
6.8 | IC50 | 3 | — | |
YFUJBCSOUCJRRP
|
6.8 | IC50 | 3 | — | |
KSKHYUVIRUJNSQ
|
6.8 | IC50 | 3 | — | |
UTEPROJRMFGHNF
|
6.8 | IC50 | 3 | — | |
FQEYESALQSIRAQ
|
6.8 | IC50 | 3 | — | |
OGFUMLMDBRBYKQ
|
6.8 | IC50 | 3 | — | |
RUPINSRFDWKDBS
|
6.8 | IC50 | 3 | — | |
UUEYTEZBJWMVIQ
|
6.8 | IC50 | 5 | Yes | |
DYTKVFHLKPDNRW
|
6.8 | Ki | 23 | Yes | |
RGUQJUZAJQPBOS
|
6.8 | IC50 | 3 | — | |
UWHYTXRXDYNHKS
|
6.8 | IC50 | 3 | — | |
JOEZGPVMIDNCJZ
|
6.8 | IC50 | 5 | Yes | |
QGLVSYZUEILELT
|
6.8 | IC50 | 3 | — | |
QMCPPBRAJKQPLH
|
6.8 | IC50 | 3 | — | |
YXTDYCAIPCZQMK
|
6.8 | IC50 | 3 | — | |
IJFFMXZETMQIDH
|
6.8 | IC50 | 3 | — | |
WJAXVXBCECPBCW
|
6.8 | IC50 | 3 | — | |
NSKYYUZMAXEZIR
|
6.7 | Ki | 15 | — | |
ZTVQNBOBFFHIID
|
6.7 | IC50 | 3 | — | |
DKZYXHCYPUVGAF
|
6.7 | Kd | 112 | — | |
AAKJLRGGTJKAMG
|
6.7 | Kd | 50 | Yes | |
YHRRFPHKXXYHDL
|
6.7 | IC50 | 5 | Yes | |
DACQLXDKBYZOIO
|
6.7 | IC50 | 3 | — | |
CHWHVQUNCYDPDK
|
6.7 | IC50 | 6 | Yes | |
INWRCUFOGIVMJS
|
6.7 | IC50 | 3 | — | |
PJGPXHUOFQXHSM
|
6.7 | IC50 | 3 | — | |
GXAIYZPLZBVGNJ
|
6.7 | IC50 | 3 | — | |
MRAGPKBXJJGPCW
|
6.7 | IC50 | 3 | — | |
XGRIDNQIXZILPG
|
6.7 | IC50 | 3 | — | |
FPPFXZVOJMZPIB
|
6.7 | IC50 | 5 | Yes | |
VEPKQEUBKLEPRA
|
6.7 | Kd | 11 | — | |
KIRQYDLDUZGZPQ
|
6.7 | IC50 | 3 | — | |
LKPYVIHIXNNVJX
|
6.7 | IC50 | 3 | — | |
QGPSFIYTQAONCS
|
6.6 | IC50 | 5 | Yes | |
VNYKLXOIIZFVQW
|
6.6 | IC50 | 5 | Yes | |
VSCYVMFGKQHZQG
|
6.6 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
BRUSFAZPHIPJRR
|
6.6 | IC50 | 5 | Yes | |
UFLGKZDFVFEGCP
|
6.6 | IC50 | 6 | Yes | |
JXOIAMLUKJBNFR
|
6.5 | IC50 | 4 | Yes | |
ZJKZZFVTJGIADM
|
6.5 | IC50 | 2 | — | |
BFSMGDJOXZAERB
|
6.5 | Kd | 33 | — | |
DYVPNYHYZSMFSR
|
6.5 | IC50 | 5 | Yes | |
RUAMUEWFVAEXLC
|
6.5 | IC50 | 3 | — | |
SPMVMDHWKHCIDT
|
6.5 | Kd | 30 | — | |
APPXQUDJLJXULP
|
6.5 | IC50 | 47 | — | |
YRCHYHRCBXNYNU
|
6.5 | Kd | 13 | — | |
JSAIPLUIDULEAD
|
6.5 | IC50 | 3 | — | |
RLICCWOKSVSSOF
|
6.5 | IC50 | 5 | Yes | |
LNMRSSIMGCDUTP
|
6.5 | Kd | 13 | — |