Target Details
| UniProt AC | P42684 |
|---|---|
| Gene Symbol | ABL2 |
| Protein Name | Tyrosine-protein kinase ABL2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 202
- Clinical molecules 75
- Avg pChEMBL 6.99
KEGG Pathways (4)
Active Molecules (202)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FYTNSFVHUFSPDY
|
7.3 | IC50 | 3 | — | |
SMFAJPHTYQUDOC
|
7.3 | IC50 | 5 | Yes | |
SWWHQLAUNHTMIH
|
7.3 | IC50 | 2 | — | |
AKRIJSSBKYPXID
|
7.3 | IC50 | 3 | — | |
RHWUJWQTWHXYPV
|
7.3 | IC50 | 3 | — | |
UMBFDGUGXMOMHX
|
7.3 | IC50 | 12 | — | |
XQKRNUCXAFMEFO
|
7.3 | IC50 | 3 | — | |
NMCRRFLWJZUPRE
|
7.3 | IC50 | 5 | Yes | |
WHGYBXFWUBPSRW
|
7.3 | Kd | 2 | — | |
HKBVCGJVIFGBEX
|
7.2 | IC50 | 6 | Yes | |
QSBWHISTPSABIV
|
7.2 | IC50 | 4 | Yes | |
DDCRNOXQNBDLGB
|
7.2 | IC50 | 4 | Yes | |
JSPJGKUIWGWCRE
|
7.2 | IC50 | 5 | Yes | |
AGENIADQYCDWLP
|
7.2 | IC50 | 3 | — | |
JXXVUIBYJYNDBA
|
7.2 | IC50 | 3 | — | |
QEKCMFKWDZHOOD
|
7.2 | IC50 | 6 | Yes | |
RITAVMQDGBJQJZ
|
7.2 | Kd | 43 | — | |
UHTHHESEBZOYNR
|
7.2 | Kd | 66 | Yes | |
SLEWGGZPOQNVSU
|
7.2 | Kd | 22 | — | |
OJOMKFBUCUYZRW
|
7.1 | IC50 | 3 | — | |
XJNQIRXYMVFKTA
|
7.1 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
SMPGEBOIKULBCT
|
7.1 | IC50 | 15 | — | |
ADGOPPKEIZXKAZ
|
7.1 | IC50 | 3 | — | |
LCVIRAZGMYMNNT
|
7.1 | Kd | 20 | — | |
NFCXPDAZPBFBRT
|
7.1 | IC50 | 3 | — | |
FRSWPGKMMGVEGT
|
7.1 | IC50 | 2 | — | |
KAUYVUREAPHUSF
|
7.1 | IC50 | 5 | Yes | |
QCUODDVWGHBDKJ
|
7.1 | IC50 | 3 | — | |
QXLGSVJYRNECIT
|
7.1 | IC50 | 3 | — | |
OVPLBDSXFCRGJY
|
7.0 | IC50 | 5 | Yes | |
SRTONYAWGLMSSN
|
7.0 | IC50 | 4 | Yes | |
OUKYUETWWIPKQR
|
7.0 | Kd | 31 | Yes | |
PKDOQGUKLRAMEF
|
7.0 | IC50 | 3 | — | |
WJSCDYSIDGEWEB
|
7.0 | IC50 | 5 | Yes | |
CAAAKLVRRGRQHX
|
7.0 | IC50 | 3 | — | |
VWMJHAFYPMOMGF
|
7.0 | Kd | 15 | — | |
YMHOIAKNPORUIV
|
7.0 | IC50 | 3 | — | |
CAMZXNIVTYLQCA
|
7.0 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 213 | — | |
PXGNDOOTUBVRMA
|
7.0 | IC50 | 5 | Yes | |
WJEOLQLKVOPQFV
|
7.0 | Kd | 24 | — | |
OBLBAQUXHOPUQG
|
6.9 | IC50 | 3 | — | |
VZSOVTDSOYVYSF
|
6.9 | IC50 | 3 | — | |
HUZDGCVNDDSQGA
|
6.9 | IC50 | 6 | Yes | |
GFNNBHLJANVSQV
|
6.9 | IC50 | 7 | Yes | |
RQMAVXSBMSSQDJ
|
6.9 | IC50 | 3 | — | |
WVXNSAVVKYZVOE
|
6.9 | Kd | 92 | — | |
UUUZEMLVABCSCR
|
6.9 | IC50 | 3 | — | |
SFSJABJVSLHBAD
|
6.8 | IC50 | 5 | Yes |