Target Details
| UniProt AC | P42684 |
|---|---|
| Gene Symbol | ABL2 |
| Protein Name | Tyrosine-protein kinase ABL2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 202
- Clinical molecules 75
- Avg pChEMBL 6.99
KEGG Pathways (4)
Active Molecules (202)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZBNZXTGUTAYRHI
|
9.8 | Kd | 102 | Yes | |
VAARYSWULJUGST
|
9.2 | Kd | 119 | Yes | |
QXWCRBMAGJJKTO
|
9.1 | IC50 | 4 | Yes | |
AQSSMEORRLJZLU
|
9.0 | Kd | 34 | Yes | |
UBPYILGKFZZVDX
|
9.0 | IC50 | 130 | Yes | |
IBRPSHUYWHRYQA
|
8.9 | IC50 | 4 | Yes | |
VSJSIOZQNZPUAV
|
8.8 | IC50 | 3 | — | |
QSECCHMWSVTBKZ
|
8.6 | IC50 | 4 | Yes | |
FCIILWHQWNLPJU
|
8.5 | IC50 | 4 | Yes | |
TXAYKQMEBQBGLR
|
8.5 | IC50 | 4 | Yes | |
ODPGGGTTYSGTGO
|
8.5 | Kd | 153 | — | |
ZPKGDYKWVKCDJQ
|
8.5 | IC50 | 4 | Yes | |
GCIKSSRWRFVXBI
|
8.4 | Kd | 109 | Yes | |
YHVHYWYQEFELOW
|
8.4 | IC50 | 44 | — | |
MXWHSGSOZDOVLL
|
8.3 | IC50 | 4 | Yes | |
ZUMNLSFJINJANM
|
8.3 | IC50 | 5 | Yes | |
WCWDBZHYAHZGNZ
|
8.3 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
8.1 | Kd | 55 | — | |
YAFBWUKWKZZPIF
|
8.1 | IC50 | 4 | Yes | |
YQWRDEHPSFGGHV
|
8.1 | IC50 | 4 | Yes | |
BLYRPGBSIKAIAU
|
8.0 | IC50 | 24 | Yes | |
XKFTZKGMDDZMJI
|
8.0 | Kd | 64 | Yes | |
ZGBAJMQHJDFTQJ
|
8.0 | Kd | 15 | — | |
MIMOHMCANSGXIG
|
8.0 | IC50 | 15 | — | |
KTUFNOKKBVMGRW
|
7.9 | Kd | 38 | Yes | |
BWLSIYJKVFXNFV
|
7.9 | IC50 | 4 | Yes | |
OZLFFPLKFGJQDT
|
7.9 | IC50 | 2 | — | |
QAZSOKNYSVTMPH
|
7.9 | IC50 | 3 | — | |
ONVKFNZGEFTWQD
|
7.8 | IC50 | 4 | Yes | |
OOMBFNDWQIGHEK
|
7.8 | Kd | 22 | — | |
KZYSNMDDKMTSHZ
|
7.8 | IC50 | 3 | — | |
SQJDLYFEJSIHPR
|
7.8 | IC50 | 2 | — | |
AFVGAHBUCVDPPI
|
7.7 | IC50 | 6 | Yes | |
PHXJVRSECIGDHY
|
7.7 | Kd | 59 | — | |
HHZIURLSWUIHRB
|
7.6 | Kd | 57 | Yes | |
SEJGTFPOEJWEGG
|
7.6 | Kd | 149 | — | |
NYKXOFIGGDPRIF
|
7.6 | IC50 | 2 | — | |
DKNUPRMJNUQNHR
|
7.5 | Kd | 33 | — | |
NWKLIKWHLFEAFY
|
7.5 | IC50 | 2 | — | |
BVQJGEBCGLWTNC
|
7.5 | IC50 | 3 | — | |
OWSMSMNEFKFQBZ
|
7.5 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.4 | Kd | 154 | — | |
YCFQNCQMGGRGHM
|
7.4 | IC50 | 4 | Yes | |
HXPKYBPDEWUZKU
|
7.4 | IC50 | 3 | — | |
CAHQAXRCSXNZRF
|
7.4 | IC50 | 5 | Yes | |
CSGQVNMSRKWUSH
|
7.4 | Kd | 21 | — | |
VISDQUKQUGPQNV
|
7.4 | IC50 | 5 | Yes | |
JVSPTGDDSIVSOE
|
7.3 | IC50 | 3 | — | |
VIHCLUIQGPQVJO
|
7.3 | IC50 | 3 | — | |
DHKJMXHLKKNTKJ
|
7.3 | IC50 | 5 | Yes |