Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRMPAHQCEQZGQI
|
6.3 | IC50 | 3 | — | |
YEZJNYHSUDDMPA
|
6.3 | IC50 | 2 | — | |
UPBLLWLBMPEKKB
|
6.2 | IC50 | 2 | — | |
XZAATUBTUPPERZ
|
6.2 | IC50 | 6 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
GKZGJDDKZTVQJZ
|
6.2 | IC50 | 4 | — | |
AUUIJHXHLCNNBO
|
6.2 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
6.2 | Kd | 289 | Yes | |
OMZCMEYTWSXEPZ
|
6.2 | Kd | 43 | Yes | |
PGENIWTWTKBDBN
|
6.2 | IC50 | 3 | — | |
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
OETOLISJTPMUFM
|
6.1 | Kd | 4 | — | |
VQUUBQYYHFHNFA
|
6.1 | IC50 | 4 | — | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
OSAWFUCUZJNEID
|
6.0 | IC50 | 20 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
NXSJMRCTGYTSTK
|
6.0 | Kd | 200 | — |