Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZLXZLDAFTMTABQ
|
6.8 | IC50 | 2 | — | |
ZXMXYLXJUSLMQW
|
6.8 | IC50 | 4 | — | |
TVJRDCQUZMGBAB
|
6.7 | IC50 | 13 | — | |
UBUVIQYWARUKMQ
|
6.7 | IC50 | 4 | — | |
NFLKTKKJFVNGLH
|
6.7 | IC50 | 4 | — | |
ZKWWEOIHGRQYDB
|
6.7 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
6.6 | Kd | 213 | — | |
LSJWYMSFUWBGPN
|
6.6 | IC50 | 17 | — | |
OPKHZFMFWCMAPS
|
6.6 | IC50 | 6 | — | |
LXMWGYNOGUKODT
|
6.6 | IC50 | 3 | — | |
LAUHLGUSVSJYCI
|
6.6 | IC50 | 16 | — | |
LUMAVJBHSUJPOG
|
6.6 | IC50 | 4 | — | |
BBDSYVIXESVDPE
|
6.6 | IC50 | 4 | — | |
GZYUJXFTHLKPAK
|
6.5 | IC50 | 16 | — | |
VYZQSAKXLMEDCB
|
6.5 | IC50 | 9 | — | |
ABSANYKJICYHQP
|
6.5 | IC50 | 4 | — | |
VRASPPLZZRUGFU
|
6.5 | IC50 | 2 | — | |
WMMNTQFZCHUZSM
|
6.5 | IC50 | 14 | — | |
MFAQYJIYDMLAIM
|
6.5 | Kd | 130 | Yes | |
RMTJSBZCZKCYHB
|
6.5 | IC50 | 13 | — | |
LXURGGKEOPHREO
|
6.5 | IC50 | 13 | — | |
CVBABGVEYUMHNU
|
6.4 | IC50 | 6 | — | |
VSFINVOSLLRTIP
|
6.4 | IC50 | 6 | — | |
WDENQIQQYWYTPO
|
6.4 | IC50 | 8 | — | |
SBGMPUIVPOGTGN
|
6.4 | Kd | 4 | — | |
RGZXAQQHXALOBL
|
6.4 | Kd | 10 | — | |
GEEUDEOZMWBPDT
|
6.4 | IC50 | 4 | — | |
YBKODNZGBUDZRA
|
6.4 | IC50 | 3 | — | |
WDTHDWKPTWWHLS
|
6.3 | IC50 | 13 | — | |
QQWUGDVOUVUTOY
|
6.3 | Kd | 231 | Yes | |
JHBYRHQSNOLZKK
|
6.3 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.3 | Kd | 149 | — | |
ZJSNZHATZAWKIQ
|
6.3 | Kd | 5 | — | |
BLXPCDKRTUJRIL
|
6.3 | IC50 | 3 | — | |
ITSFNGBRTUQMRR
|
6.3 | IC50 | 2 | — | |
JLYFULJVYPGNKH
|
6.3 | IC50 | 2 | — | |
KGDQFYISJYCDCR
|
6.3 | IC50 | 3 | — | |
KJMXXXANAMPTLR
|
6.3 | IC50 | 3 | — | |
MVLQRJLRLWTRKD
|
6.3 | IC50 | 2 | — | |
MZEUUPBYZLOHJY
|
6.3 | IC50 | 3 | — | |
NCRMRUFKSNRKJO
|
6.3 | IC50 | 4 | — | |
NPLQEGUXLSILFV
|
6.3 | IC50 | 3 | — | |
ONKCBNMZBWUKKB
|
6.3 | IC50 | 3 | — | |
PUQQULIZFUPRHD
|
6.3 | IC50 | 3 | — | |
TWEWIWWUVQHFTP
|
6.3 | IC50 | 2 | — | |
UMJITRWVLLDKIH
|
6.3 | IC50 | 2 | — | |
XAYYFPBZEBIJJN
|
6.3 | IC50 | 2 | — | |
XEJWPSGQNGGXNI
|
6.3 | IC50 | 2 | — | |
XIXSOBAWBJNKQI
|
6.3 | IC50 | 3 | — |