Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QRIXKWMQRHCONV
|
6.9 | IC50 | 4 | — | |
SDVAHCXGDGYWFA
|
6.9 | IC50 | 12 | — | |
ATLOUNJJIAISOI
|
6.9 | IC50 | 4 | — | |
VTJHGMZHVOXJPG
|
6.9 | IC50 | 15 | — | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
NMNLVTJEQAQJHN
|
6.8 | IC50 | 4 | — | |
WZLCFQWCRHXUJG
|
6.8 | IC50 | 4 | — | |
CBRJPFGIXUFMTM
|
6.8 | IC50 | 7 | — | |
FTWCGCABDYPPKS
|
6.8 | IC50 | 4 | — | |
BQOLJLKHTXMXTC
|
6.8 | IC50 | 3 | — | |
CGQNXESNFIWIFE
|
6.8 | IC50 | 3 | — | |
CIXVBIGXYDABFE
|
6.8 | IC50 | 3 | — | |
CLBPSWFERFXVHT
|
6.8 | IC50 | 3 | — | |
CTMYBLAMYVZJHP
|
6.8 | IC50 | 2 | — | |
CUYLWVQYAWJAJO
|
6.8 | IC50 | 4 | — | |
CWNRVQNBVZMOTJ
|
6.8 | IC50 | 3 | — | |
DEIVZTMEKYQXQT
|
6.8 | IC50 | 3 | — | |
DMVHLNHVYRCQEH
|
6.8 | IC50 | 3 | — | |
FFNUJLRFLYSCQK
|
6.8 | IC50 | 3 | — | |
FKRLXQSJKAMNDA
|
6.8 | IC50 | 3 | — | |
FVVMFZQDPMKOCB
|
6.8 | IC50 | 3 | — | |
HCZWFMCFNBYKCL
|
6.8 | IC50 | 4 | — | |
IEYVQQYVGOEFOU
|
6.8 | IC50 | 3 | — | |
IWEOUDKFSYHECW
|
6.8 | IC50 | 3 | — | |
JOLPRIOSDDVVTE
|
6.8 | IC50 | 3 | — | |
KNCWSXRTKLTULH
|
6.8 | IC50 | 4 | — | |
KNCWSXRTKLTULH
|
6.8 | IC50 | 3 | — | |
KNSUJTHSBPKFCJ
|
6.8 | IC50 | 3 | — | |
KUCKLOIPORVHKG
|
6.8 | IC50 | 3 | — | |
KYICFMVZOZDKNA
|
6.8 | IC50 | 3 | — | |
LGDMBUJSUZUYOR
|
6.8 | IC50 | 3 | — | |
LIQTYBXZDKCJCT
|
6.8 | IC50 | 4 | — | |
MASQAZICCWGIQC
|
6.8 | IC50 | 4 | — | |
NTWLRXFMUQKCDK
|
6.8 | IC50 | 3 | — | |
OLKAUBUUBHWFHE
|
6.8 | IC50 | 3 | — | |
OQMMZZSWHUDPHF
|
6.8 | IC50 | 3 | — | |
RETXECLWCXMDDQ
|
6.8 | IC50 | 4 | — | |
RMKSFFNCKQXFNQ
|
6.8 | IC50 | 2 | — | |
ROXFXAIVSYHQLR
|
6.8 | IC50 | 3 | — | |
SEHHTFNWOYVBEW
|
6.8 | IC50 | 3 | — | |
SGSHTWFWXWRCJJ
|
6.8 | IC50 | 3 | — | |
SHLOWQBVNWTKOE
|
6.8 | IC50 | 4 | — | |
SHLOWQBVNWTKOE
|
6.8 | IC50 | 3 | — | |
SVGNRMVKDQYWFL
|
6.8 | IC50 | 3 | — | |
UMBDWDIRLTVPBF
|
6.8 | IC50 | 9 | — | |
UQQGDOHGERGPIF
|
6.8 | IC50 | 3 | — | |
VSVMYZKXQYJROQ
|
6.8 | IC50 | 3 | — | |
XWUWNWYEAQWLAL
|
6.8 | IC50 | 3 | — | |
XZLNPOIHGOJYFH
|
6.8 | IC50 | 3 | — | |
YVTVSMGMGCBOKG
|
6.8 | IC50 | 3 | — |