Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GFZZUAFZBKEOHV
|
7.6 | IC50 | 7 | — | |
CLKNHJDZJCCLAZ
|
7.6 | IC50 | 4 | — | |
ADCQRIVAZWFZCZ
|
7.5 | IC50 | 4 | — | |
ZRYMMWAJAFUANM
|
7.5 | IC50 | 7 | — | |
WJYODWGPCZGFIM
|
7.5 | IC50 | 2 | — | |
XYFZVVYVIFJBIS
|
7.5 | IC50 | 17 | — | |
JUSWPUDQOKINJO
|
7.5 | IC50 | 16 | — | |
SRSQULBCTWSVKL
|
7.5 | IC50 | 15 | — | |
AHGUJKCTSXOYES
|
7.5 | IC50 | 4 | — | |
HJAUUHMYFPHMCT
|
7.5 | IC50 | 4 | — | |
VAARYSWULJUGST
|
7.5 | Kd | 119 | Yes | |
UGXCBYVBIJACEK
|
7.4 | IC50 | 8 | — | |
BPMZEUVOCIAUDQ
|
7.4 | IC50 | 4 | — | |
ZZJOFPXLPFXEKV
|
7.4 | IC50 | 4 | — | |
NZIQNLGMMJGSQU
|
7.3 | IC50 | 6 | — | |
OPHSZSZDICRBPP
|
7.3 | IC50 | 16 | — | |
CDISOBGWDHAHGF
|
7.3 | IC50 | 16 | — | |
SXLIACXIXLLKGR
|
7.3 | IC50 | 4 | — | |
AHBFBRPGNOVEBK
|
7.3 | IC50 | 11 | — | |
DNFWTELNLRENAM
|
7.3 | IC50 | 4 | — | |
YCPPFUIKNAOWRT
|
7.3 | IC50 | 3 | — | |
CMFVTAHMZDUCJB
|
7.3 | IC50 | 10 | — | |
UBPYILGKFZZVDX
|
7.3 | IC50 | 130 | Yes | |
IGXJXMLDIIGDNE
|
7.3 | IC50 | 8 | — | |
YYRYNQBAVOOSOA
|
7.3 | IC50 | 4 | — | |
PVCKRSKEOOWVMP
|
7.2 | IC50 | 4 | — | |
DNDCQFCAXLONFM
|
7.2 | IC50 | 4 | — | |
VPBAASZNSPZLLC
|
7.2 | IC50 | 2 | — | |
CZSSHLOWZFKWML
|
7.2 | IC50 | 3 | — | |
YMGVIVNBLOXKBY
|
7.2 | IC50 | 2 | — | |
OHAIFZDRLDEOAC
|
7.2 | IC50 | 3 | — | |
HDVYJNSAOAUAIQ
|
7.2 | IC50 | 4 | — | |
RJARQSDFMBQVEH
|
7.2 | IC50 | 4 | — | |
FVSUKLKFSDSIEF
|
7.1 | IC50 | 4 | — | |
CQZZZUNOWZUNNG
|
7.1 | IC50 | 4 | — | |
QNNJMWIVIVLSHC
|
7.1 | IC50 | 4 | — | |
CIGMIXWAESLRNR
|
7.1 | Kd | 5 | — | |
DOVHWPFJHQGYDS
|
7.1 | IC50 | 4 | — | |
DPRNXTSMYVCYLJ
|
7.1 | IC50 | 13 | — | |
ZXGCNNKDPNECIS
|
7.1 | IC50 | 4 | — | |
GAWQIOVCXHLEAP
|
7.1 | Kd | 4 | — | |
ZYQIUDPJBOUHCC
|
7.0 | IC50 | 4 | — | |
KOQJXUXLQGQJDF
|
7.0 | IC50 | 4 | — | |
YPXWUKLQAUBCPF
|
7.0 | IC50 | 8 | — | |
KQISOZQPFQHIFH
|
7.0 | IC50 | 4 | — | |
KRILZVCKKUOPKH
|
7.0 | IC50 | 4 | — | |
OMIQRSKHABIPRH
|
7.0 | IC50 | 15 | — | |
WCCLANJGOUJNNL
|
7.0 | IC50 | 4 | — | |
SEJLPXCPMNSRAM
|
6.9 | IC50 | 7 | — | |
BLOSAGLLXHJECN
|
6.9 | IC50 | 4 | — |