Target Details
| UniProt AC | P42681 |
|---|---|
| Gene Symbol | TXK |
| Protein Name | Tyrosine-protein kinase TXK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 419
- Clinical molecules 8
- Avg pChEMBL 7.88
KEGG Pathways (1)
Active Molecules (419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KAFKHBRCDYVZDT
|
8.5 | IC50 | 4 | — | |
KZMQPYCXSAGLTB
|
8.5 | IC50 | 8 | — | |
ZFDGMDVYMNWICG
|
8.5 | IC50 | 10 | — | |
FQYPYAFBYPJBLZ
|
8.5 | IC50 | 2 | — | |
BUXSSQZWDXOIAY
|
8.4 | IC50 | 2 | — | |
FINZRTUQZUBKBD
|
8.4 | IC50 | 3 | — | |
SXXABOHFQFARBT
|
8.4 | IC50 | 5 | — | |
DQFOPMWZUFUHDC
|
8.4 | IC50 | 6 | — | |
OYFVJVWLUDKTIF
|
8.4 | IC50 | 4 | — | |
MRNPOLZRBHNDGI
|
8.4 | IC50 | 4 | — | |
AOKKWYGSIRAXIZ
|
8.3 | IC50 | 4 | — | |
VWJGTQUINXNBOY
|
8.3 | IC50 | 4 | — | |
VJPPLCNBDLZIFG
|
8.3 | IC50 | 5 | — | |
CKXVUTSXVABAMG
|
8.3 | IC50 | 4 | — | |
FKBBYUQWEWBQAS
|
8.3 | IC50 | 2 | — | |
BGGDZMOTNWYYKG
|
8.2 | IC50 | 2 | — | |
HFGNFXUUAVQOCF
|
8.2 | IC50 | 2 | — | |
YHVHYWYQEFELOW
|
8.2 | IC50 | 44 | — | |
SUHPRCQYTXOSRF
|
8.2 | IC50 | 4 | — | |
CDFHNEWIEMNZKE
|
8.2 | IC50 | 4 | — | |
MOQPPOYWQCSUFS
|
8.1 | IC50 | 2 | — | |
JKTAWSRABQDLCF
|
8.1 | IC50 | 2 | — | |
XNPHXLCYBBQUQK
|
8.1 | IC50 | 4 | — | |
VYVIHHSHQWYIAI
|
8.1 | IC50 | 3 | — | |
NUDBRCUXDGGUOA
|
8.1 | IC50 | 4 | — | |
CDUYTHAOJIKLFN
|
8.0 | IC50 | 4 | — | |
NAXFVNQSUIOSIC
|
8.0 | IC50 | 4 | — | |
PYCLWFJRXCZMNR
|
8.0 | IC50 | 2 | — | |
IRBVGTPPFBYDKX
|
8.0 | IC50 | 9 | — | |
SFCBIFOAGRZJNX
|
8.0 | Kd | 22 | — | |
FMRJPPUXBYSJRE
|
8.0 | IC50 | 4 | — | |
UQPCMSBCSBHRAK
|
8.0 | IC50 | 3 | — | |
MNDLPZPZVIEBFF
|
7.9 | IC50 | 4 | — | |
UVUTZINLTAEGAD
|
7.9 | IC50 | 4 | — | |
LHLGYQRKVKDWSY
|
7.8 | IC50 | 4 | — | |
XIDJFSRGLOUDGG
|
7.8 | IC50 | 4 | — | |
FUZSHLVNKZZEKR
|
7.8 | IC50 | 16 | — | |
QCJFYACTZIVZBB
|
7.8 | IC50 | 8 | — | |
SBRIQINKAOKMMM
|
7.8 | IC50 | 6 | — | |
IZQVCAWYZWMWJS
|
7.8 | IC50 | 4 | — | |
AAXRDDUUPKFSOA
|
7.8 | IC50 | 3 | — | |
AJPQBQFAMSEUAN
|
7.8 | IC50 | 3 | — | |
AZSVIPLAHQKWFG
|
7.8 | IC50 | 3 | — | |
BAHKFTMIURNVFB
|
7.8 | IC50 | 3 | — | |
CECVIWNNFCTJPO
|
7.8 | IC50 | 4 | — | |
DIDSIJOVKDQRQB
|
7.8 | IC50 | 3 | — | |
DXPSTMYIXNPVBW
|
7.8 | IC50 | 3 | — | |
DZIBWEFMBVZGAL
|
7.8 | IC50 | 3 | — | |
FTVAMBICGBZUSH
|
7.8 | IC50 | 3 | — | |
FWZAVTIYCKNCTE
|
7.8 | IC50 | 3 | — |